SCHEMBL11150271

SCHEMBL11150271

CC(=O)OCCn1c(=O)c2cc3c(=O)n(C(C)=O)c(=O)c3cc2c1=O

nearest known ligand 0.84

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.84
GAA P10253 3/20 0.60
POLB P06746 1/20 0.59
NPSR1 Q6W5P4 1/20 0.59
ADORA2B P29275 2/20 0.49
KDM4E B2RXH2 4/20 0.46
MAPT P10636 3/20 0.39
RXFP1 Q9HBX9 2/20 0.38
HTT P42858 2/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
IDO1 P14902 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
SLC18A3 Q16572 1/20 0.37
TP53 P04637 1/20 0.35
MAPK1 P28482 1/20 0.35
PARG Q86W56 1/20 0.35
PTGS2 P35354 1/20 0.34
APOBEC3A P31941 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11152031 0.83 ALDH1A1 (0.82) ALDH1A1GAAPOLBNPSR1ADORA2B
SCHEMBL11151949 0.80 ALDH1A1 (0.53) ALDH1A1GAAPOLBNPSR1ADORA2B
SCHEMBL13863953 0.78 ALDH1A1 (0.73) ALDH1A1GAAPOLBNPSR1ADORA2B
SCHEMBL11266479 0.74 ALDH1A1 (0.68) ALDH1A1GAAPOLBNPSR1ADORA2B
SCHEMBL24439270 0.74 ALDH1A1 (0.51) ALDH1A1GAAPOLBNPSR1KDM4E
SCHEMBL1729796 0.71 ALDH1A1 (0.64) ALDH1A1GAAPOLBNPSR1ADORA2B
SCHEMBL29674700 0.71 NPC1 (0.49) ALDH1A1GAAPOLBNPSR1MAPT
SCHEMBL13863955 0.70 KDM4E (0.61) ALDH1A1GAAPOLBNPSR1ADORA2B
SCHEMBL24439007 0.70 ALDH1A1 (0.42) ALDH1A1GAAPOLBNPSR1
SCHEMBL13863951 0.70 KDM4E (0.61) ALDH1A1GAAPOLBNPSR1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0010440-B1 PYROMELLITIC DIIMIDES, PROCESSES FOR THEIR PREPARATION, THESE COMPOUNDS IN ORALLY ADMINISTRABLE FORM FOR USE IN INCREASING THE FEED EFFICIENCY OF A RUMINANT ANIMAL AND COMPOSITIONS FOR THIS PURPOSE CONTAINING THEM MERCK & CO. INC. (US) 1983-01-26 EP disclosed
US-4289784-A ASYMMETRICALLY SUBSTITUTED MERCK & CO., INC. (US) 1981-09-15 US disclosed
EP-0010440-A1 Pyromellitic diimides, processes for their preparation, these compounds in orally administrable form for use in increasing the feed efficiency of a ruminant animal and compositions for this purpose containing them MERCK & CO. INC. (US) 1980-04-30 EP disclosed