SCHEMBL11154239

SCHEMBL11154239

O=C1c2ccccc2OC12CC2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
PPIB P23284 1/20 0.43
TSHR P16473 2/20 0.41
PKM P14618 1/20 0.41
ATM Q13315 1/20 0.40
MAPT P10636 2/20 0.39
HPGD P15428 2/20 0.39
SIGMAR1 Q99720 1/20 0.38
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
HDAC3 O15379 3/20 0.37
HDAC4 P56524 3/20 0.37
HDAC1 Q13547 3/20 0.37
HDAC7 Q8WUI4 3/20 0.37
HDAC2 Q92769 3/20 0.37
HDAC10 Q969S8 3/20 0.37
HDAC11 Q96DB2 3/20 0.37
HDAC8 Q9BY41 3/20 0.37
HDAC6 Q9UBN7 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28202516 0.92 ALDH1A1 (0.47) ALDH1A1PPIBTSHRPKMATM
SCHEMBL27587 0.90 ALDH1A1 (0.54) ALDH1A1PPIBTSHRPKMATM
SCHEMBL10603717 0.90 ALDH1A1 (0.54) ALDH1A1PPIBTSHRPKMATM
SCHEMBL3110019 0.89 ALDH1A1 (0.41) ALDH1A1PPIBTSHRPKMATM
SCHEMBL22389768 0.87 HDAC3 (0.50) ALDH1A1SIGMAR1HDAC3HDAC4HDAC1
Hydrochloric Acid SCHEMBL3228756 0.86 HDAC3 (0.49) ALDH1A1SIGMAR1HDAC3HDAC4HDAC1
SCHEMBL21037722 0.84 HDAC3 (0.51) PPIBSIGMAR1HDAC3HDAC4HDAC1
SCHEMBL21037721 0.81 CYP2D6 (0.44) ALDH1A1PPIBMAPTSIGMAR1HDAC3
SCHEMBL21383845 0.81 HDAC3 (0.48) SIGMAR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL28549888 0.77 HDAC3 (0.43) PPIBSIGMAR1HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0003084-B1 SPIROBENZOFURANONE COMPOUNDS, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS MEDICINES Takeda Chemical Industries, Ltd. (JP) 1982-02-24 EP claimed
US-4284644-A Spirobenzofuranone compounds TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1981-08-18 US claimed
JP-55064582-A None JP disclosed
JP-56005473-A None JP disclosed
JP-54098752-A None JP disclosed
EP-0018830-B1 SPIROBENZOFURANONES, THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Takeda Chemical Industries, Ltd. (JP) 1983-06-08 EP disclosed
EP-0003084-B1 SPIROBENZOFURANONE COMPOUNDS, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS MEDICINES Takeda Chemical Industries, Ltd. (JP) 1982-02-24 EP disclosed
JP-S565473-A SPIRO COMPOUND AND ITS PREPARATION TAKEDA CHEM IND LTD 1981-01-20 JP disclosed
EP-0018830-A2 Spirobenzofuranones, their production and pharmaceutical compositions containing them Takeda Chemical Industries, Ltd. (JP) 1980-11-12 EP disclosed
JP-S5564582-A SPIRO COMPOUND AND ITS PREPARATION TAKEDA CHEM IND LTD 1980-05-15 JP disclosed
JP-S5498752-A SPIRO COMPOUND AND ITS PREPARATION TAKEDA CHEM IND LTD 1979-08-03 JP disclosed
EP-0003084-A1 Spirobenzofuranone compounds, processes for their preparation and their use as medicines Takeda Chemical Industries, Ltd. (JP) 1979-07-25 EP disclosed