SCHEMBL11161069

SCHEMBL11161069

CC(N)=C(C#N)C(=O)c1ccc(F)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK10 P53779 2/20 0.53
TP53 P04637 1/20 0.53
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
ALDH1A1 P00352 6/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
TDP1 Q9NUW8 4/20 0.43
RAB9A P51151 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
NPC1 O15118 1/20 0.43
LMNA P02545 3/20 0.42
MAPK1 P28482 2/20 0.42
MAPT P10636 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
XBP1 P17861 1/20 0.42
TSHR P16473 1/20 0.41
KCNH2 Q12809 1/20 0.41
EGFR P00533 1/20 0.41
ERBB2 P04626 1/20 0.41
ALPG P10696 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11161062 1.00 MAPK10 (0.53) MAPK10TP53CES2CES1ALDH1A1
SCHEMBL11330511 0.84 CES2 (0.52) MAPK10TP53CES2CES1ALDH1A1
SCHEMBL11330505 0.84 CES2 (0.52) MAPK10TP53CES2CES1ALDH1A1
SCHEMBL11341677 0.84 CES2 (0.52) MAPK10TP53CES2CES1ALDH1A1
SCHEMBL11164430 0.80 CES2 (0.47) MAPK10TP53CES2CES1ALDH1A1
SCHEMBL11164427 0.80 CES2 (0.47) MAPK10TP53CES2CES1ALDH1A1
SCHEMBL11168628 0.80 MAPK10 (0.50) MAPK10TP53CES2CES1ALDH1A1
SCHEMBL11168632 0.80 MAPK10 (0.50) MAPK10TP53CES2CES1ALDH1A1
SCHEMBL11168327 0.80 CES2 (0.47) MAPK10TP53CES2CES1ALDH1A1
SCHEMBL11367065 0.80 CES2 (0.47) MAPK10TP53CES2CES1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0035284-B1 NOVEL 2-BENZOYL-3-SUBSTITUTED-2-ALKENONITRILES AND PROCESS FOR THEIR PREPARATION AMERICAN CYANAMID COMPANY (US) 1983-07-13 EP disclosed
EP-0016277-B1 2-CARBONYL-3-HYDROXY-ALKENONITRILES, THEIR USE AS ANTI-ARTHRITIC AGENTS AND PROCESSES FOR THEIR PREPARATION AMERICAN CYANAMID COMPANY (US) 1981-12-02 EP disclosed
EP-0035284-A2 Novel 2-benzoyl-3-substituted-2-alkenonitriles and process for their preparation AMERICAN CYANAMID COMPANY (US) 1981-09-09 EP disclosed
EP-0016277-A1 2-Carbonyl-3-hydroxy-alkenonitriles, their use as anti-arthritic agents and processes for their preparation AMERICAN CYANAMID COMPANY (US) 1980-10-01 EP disclosed
WO-1980000964-A1 ANTI-INFLAMMATORY AGENTS INCLUDING 2-CARBONYL-3-HYDROXY-2-ALKENONITRILES AMERICAN CYANAMID CO (US) 1980-05-15 WO disclosed
US-4173650-A ANTIARTHRITIC AGENTS AMERICAN CYANAMID COMPANY (US) 1979-11-06 US disclosed