SCHEMBL11167697

SCHEMBL11167697

O=C(O)[C@@H]1Cc2ccc([N+](=O)[O-])cc2CN1

nearest known ligand 0.63

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PNMT P11086 12/20 0.63
ADRA2A P08913 7/20 0.63
ADRA2B P18089 3/20 0.63
ADRA2C P18825 3/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1491483 1.00 PNMT (0.63) PNMTADRA2AADRA2BADRA2C
SCHEMBL6391507 1.00 PNMT (0.63) PNMTADRA2AADRA2BADRA2C
SCHEMBL1491480 1.00 PNMT (0.63) PNMTADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL8488582 0.99 PNMT (0.62) PNMTADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL28292450 0.99 PNMT (0.62) PNMTADRA2AADRA2BADRA2C
SCHEMBL15623045 0.94 PNMT (0.56) PNMTADRA2AADRA2BADRA2C
SCHEMBL6921990 0.84 PNMT (0.61) PNMTADRA2AADRA2BADRA2C
SCHEMBL1202143 0.84 PNMT (0.61) PNMTADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL6398473 0.83 PNMT (0.60) PNMTADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL2081344 0.83 PNMT (0.60) PNMTADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0018104-B1 TETRAHYDROISOQUINOLINES, THEIR PRODUCTION AND THE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FOR USE IN THE PREVENTION OR TREATMENT OF HYPERTENSION Takeda Chemical Industries, Ltd. (JP) 1983-05-25 EP disclosed
EP-0018104-A2 Tetrahydroisoquinolines, their production and the compounds and pharmaceutical compositions containing them for use in the prevention or treatment of hypertension Takeda Chemical Industries, Ltd. (JP) 1980-10-29 EP disclosed