SCHEMBL11196364

SCHEMBL11196364

O=c1[nH]c2cc(Cl)ccc2n1CCCN1CCN(C(c2ccc(F)cc2)c2ccc(F)cc2)CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.61
CYP1A2 P05177 3/20 0.61
CYP2D6 P10635 3/20 0.61
ADRA1A P35348 3/20 0.61
DRD2 P14416 3/20 0.61
MEN1 O00255 2/20 0.61
NR1I2 O75469 2/20 0.61
LMNA P02545 2/20 0.61
CYP3A4 P08684 2/20 0.61
ADORA3 P0DMS8 2/20 0.61
ADRA2C P18825 2/20 0.61
SLC6A2 P23975 2/20 0.61
HTR2A P28223 2/20 0.61
HTR2C P28335 2/20 0.61
SLC6A4 P31645 2/20 0.61
HRH1 P35367 2/20 0.61
OPRM1 P35372 2/20 0.61
DRD3 P35462 2/20 0.61
OPRK1 P41145 2/20 0.61
PMP22 Q01453 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL11201943 0.91 P2RX7 (0.60) P2RX7CYP1A2CYP2D6ADRA1ADRD2
SCHEMBL11201875 0.90 P2RX7 (0.77) P2RX7CYP1A2CYP2D6ADRA1ADRD2
SCHEMBL1152607 0.85 P2RX7 (0.83) P2RX7CYP1A2CYP2D6ADRA1ADRD2
SCHEMBL11197906 0.85 P2RX7 (0.64) P2RX7CYP1A2CYP2D6ADRA1ADRD2
SCHEMBL1153001 0.84 P2RX7 (0.88) P2RX7CYP1A2CYP2D6ADRA1ADRD2
SCHEMBL1152704 0.83 P2RX7 (0.83) P2RX7CYP1A2CYP2D6ADRA1ADRD2
SCHEMBL11192067 0.83 P2RX7 (0.76) P2RX7CYP1A2CYP2D6ADRA1ADRD2
SCHEMBL11201448 0.83 P2RX7 (0.83) P2RX7CYP1A2CYP2D6ADRA1ADRD2
SCHEMBL1152747 0.82 P2RX7 (0.84) P2RX7CYP1A2CYP2D6ADRA1ADRD2
Hydrochloric Acid SCHEMBL11205596 0.82 P2RX7 (0.82) P2RX7CYP1A2CYP2D6ADRA1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4377578-A ANTIANAPHYLACTIC AGENTS, ANTIHISTAMINES JANSSEN PHARMACEUTICA, N.V. (BE) 1983-03-22 US disclosed
US-4250176-A BENZIMIDAZOLE-2-ONE, BENZOTHIAZOL-2-ONE, OR BENZOXAZOL-2-ONE SUBSTITUTIONS, ANTIANAPHALACTIC AGENTS, ANTIHISTAMINES JANSSEN PHARMACEUTICA N.V. (BE) 1981-02-10 US disclosed
US-4200641-A ANTIANAPHYLACTIC AGENTS, ANTIHISTAMINES JANSSEN PHARMACEUTICA, N.V. (BE) 1980-04-29 US disclosed