SCHEMBL11201497

SCHEMBL11201497

c1cc(CN2CCCC2)ccc1CN1CCCC1

nearest known ligand 0.94

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.94
HRH4 Q9H3N8 1/20 0.81
ALDH1A1 P00352 4/20 0.77
KDM4E B2RXH2 2/20 0.77
MBTD1 Q05BQ5 1/20 0.74
L3MBTL3 Q96JM7 1/20 0.74
L3MBTL1 Q9Y468 1/20 0.74
CYP2D6 P10635 1/20 0.71
CYP2C19 P33261 1/20 0.71
NCF1 P14598 1/20 0.68
CXCR4 P61073 2/20 0.67
POLB P06746 1/20 0.65
SMN1; SMN2 Q16637 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11196296 0.97 HRH3 (0.90) HRH3HRH4ALDH1A1KDM4EMBTD1
SCHEMBL4277270 0.97 HRH3 (1.00) HRH3HRH4ALDH1A1KDM4EMBTD1
Hydrochloric Acid SCHEMBL7468055 0.95 HRH3 (0.95) HRH3HRH4ALDH1A1KDM4EMBTD1
SCHEMBL6057527 0.92 HRH3 (0.81) HRH3HRH4ALDH1A1KDM4EMBTD1
SCHEMBL7937990 0.90 ALDH1A1 (0.95) HRH3HRH4ALDH1A1KDM4EMBTD1
SCHEMBL6057453 0.90 HRH3 (0.77) HRH3HRH4ALDH1A1KDM4EMBTD1
SCHEMBL2250410 0.88 HRH3 (0.74) HRH3HRH4ALDH1A1KDM4EMBTD1
Hydrochloric Acid SCHEMBL2334519 0.88 HRH3 (0.74) HRH3HRH4ALDH1A1KDM4EMBTD1
SCHEMBL22711410 0.88 HRH3 (0.74) HRH3HRH4ALDH1A1KDM4EMBTD1
SCHEMBL1276590 0.88 ALDH1A1 (1.00) HRH3HRH4ALDH1A1KDM4EMBTD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117820255-A Application of catalyst and degradation method of ester substance 上海科技大学 2024-04-05 CN disclosed
US-11517565-B2 Bis-amines, compositions, and uses related to CXCR4 inhibition EMORY UNIVERSITY (US) 2022-12-06 US disclosed
US-20200316040-A1 Bis-amines, Compositions, and Uses Related to CXCR4 Inhibition UNIV EMORY (US) 2020-10-08 US disclosed
US-10709697-B2 Bis-amines, compositions, and uses related to CXCR4 inhibition EMORY UNIVERSITY (US) 2020-07-14 US disclosed
US-20190008840-A1 Bis-amines, Compositions, and Uses Related to CXCR4 Inhibition NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2019-01-10 US disclosed
US-4414220-A HUPOGLYCEMIC, ANTIDIABETIC PFIZER INC. (US) 1983-11-08 US disclosed
US-4333932-A DIHYDROISOINDOLES, HYPOGLYCEMIC, ANTIDIABETIC PFIZER INC. (US) 1982-06-08 US disclosed
EP-0010896-B1 ORGANIC DIAMINE COMPOUNDS FOR USE AS ORAL HYPOGLYCEMIC AGENTS AND PHARMACEUTICAL COMPOSITIONS THEREOF PFIZER INC. (US) 1981-12-30 EP disclosed
US-4220650-A HYPOGLYCEMIC PFIZER INC. (US) 1980-09-02 US disclosed
EP-0010896-A1 Organic diamine compounds for use as oral hypoglycemic agents and pharmaceutical compositions thereof PFIZER INC. (US) 1980-05-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11517565-B2 Bis-amines, compositions, and uses related to CXCR4 inhibition CXCR4, CXCL12, CXCR2 HRH3 243/4885HRH4 531/4885ALDH1A1 453/4885
US-20200316040-A1 Bis-amines, Compositions, and Uses Related to CXCR4 Inhibition CXCR4, CXCL12, CXCR2 HRH3 243/4885HRH4 531/4885ALDH1A1 453/4885
US-10709697-B2 Bis-amines, compositions, and uses related to CXCR4 inhibition CXCR4, CXCL12, CXCR2 HRH3 246/4885HRH4 514/4885ALDH1A1 447/4885
US-20190008840-A1 Bis-amines, Compositions, and Uses Related to CXCR4 Inhibition CXCR4, CXCL12, CXCR2 HRH3 246/4885HRH4 514/4885ALDH1A1 447/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.