SCHEMBL11206117

SCHEMBL11206117

C[C@H](C[C@@H](C)C(=O)N1c2ccccc2C[C@@H]1OC(=O)O)C(=O)OCC(=O)OC1CC2CCC1(C)C2(C)C

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.40
CYP2C19 P33261 1/20 0.40
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10879974 0.90 CYP19A1 (0.40) CYP19A1CYP2C19
SCHEMBL11240205 0.90 ACE (0.47) CYP19A1CYP2C19
SCHEMBL10817392 0.90 ACE (0.48)
SCHEMBL11088900 0.90 ACE (0.48)
SCHEMBL10818819 0.87 CYP19A1 (0.40) CYP19A1
SCHEMBL11080471 0.85 ACE (0.43)
SCHEMBL10880216 0.79 CYP19A1 (0.40) CYP19A1CYP2C19ALDH1A1LMNA
SCHEMBL10811706 0.79 CYP19A1 (0.51) CYP19A1CYP2C19ALDH1A1LMNA
SCHEMBL10647022 0.77 ACE (0.47)
SCHEMBL10818844 0.76 ALDH1A1 (0.53) CYP19A1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0093084-A1 1-Carboxyalkanoylindoline-2-carboxylic-acid esters, their preparation, pharmaceutical compositions containing them, and their therapeutic use CIBA-GEIGY AG (CH) 1983-11-02 EP disclosed