SCHEMBL11206253

SCHEMBL11206253

COc1ccc(COC(=O)OC(=O)CN)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
IDO1 P14902 2/20 0.47
AGXT P21549 2/20 0.47
HTT P42858 2/20 0.46
MAPT P10636 1/20 0.46
NPC1 O15118 1/20 0.45
POLB P06746 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
MAOB P27338 1/20 0.45
KMT2A Q03164 2/20 0.45
MMP9 P14780 2/20 0.45
MMP1 P03956 1/20 0.45
MMP2 P08253 1/20 0.44
MMP12 P39900 1/20 0.44
TAAR1 Q96RJ0 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
FFAR1 O14842 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8830893 0.87 ALDH1A1 (0.54) ALDH1A1IDO1AGXTHTTMAPT
SCHEMBL6366124 0.87 ALDH1A1 (0.57) ALDH1A1IDO1AGXTHTTMAPT
Hydrochloric Acid SCHEMBL9312987 0.85 IDO1 (0.55) ALDH1A1IDO1AGXTHTTMAPT
SCHEMBL292834 0.83 ALDH1A1 (0.60) ALDH1A1IDO1AGXTHTTMAPT
SCHEMBL19514755 0.81 ALDH1A1 (0.51) ALDH1A1IDO1AGXTHTTMAPT
SCHEMBL2793142 0.80 ALDH1A1 (0.55) ALDH1A1KMT2A
SCHEMBL697621 0.80 ALDH1A1 (0.61) ALDH1A1IDO1AGXTHTTMAPT
SCHEMBL19514752 0.79 ALDH1A1 (0.50) ALDH1A1IDO1AGXTHTTMAPT
SCHEMBL819435 0.78 ALDH1A1 (0.55) ALDH1A1IDO1AGXTHTTNPC1
SCHEMBL6374290 0.78 ALDH1A1 (0.46) ALDH1A1IDO1AGXTHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0014437-B1 NOVEL 1-ARYL-2-ACYLAMIDO-3-FLUORO-1-PROPANOLS, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SCHERING CORPORATION (US) 1983-02-23 EP disclosed
US-4361557-A 1-Aryl-2-acylamido-3-fluoro-1-propanol acylates, methods for their use as anti-bacterial agents and compositions useful therefor SCHERING CORPORATION (US) 1982-11-30 US disclosed
US-4311857-A 1-Aryl-2-acylamido-3-fluoro-1-propanol acylates, methods for their manufacture and intermediates useful therein, methods for their use as antibacterial agents and compositions useful therefor SCHERING CORPORATION (US) 1982-01-19 US disclosed
EP-0014437-A2 Novel 1-aryl-2-acylamido-3-fluoro-1-propanols, their preparation and pharmaceutical compositions containing them SCHERING CORPORATION (US) 1980-08-20 EP disclosed