SCHEMBL11206366

SCHEMBL11206366

CNc1nc(N2CCNCC2)nc2scc(C(C)C)c12

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HTR2C P28335 1/20 0.39
KHK P50053 2/20 0.38
HRH1 P35367 1/20 0.36
ESR1 P03372 1/20 0.35
USP2 O75604 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CASP1 P29466 1/20 0.35
CASP4 P49662 1/20 0.35
CASP5 P51878 1/20 0.35
HRH4 Q9H3N8 1/20 0.34
PRKCI P41743 1/20 0.34
TSHR P16473 1/20 0.34
FLT3 P36888 1/20 0.34
P2RX3 P56373 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11202845 0.99 HTR2A (0.39) HTR2AKDM4EALDH1A1HTR2CKHK
SCHEMBL11201445 0.84 ESR1 (0.41) HTR2AKDM4EALDH1A1HTR2CKHK
SCHEMBL11200114 0.84 PRKCI (0.46) HTR2AKDM4EALDH1A1HTR2CKHK
Hydrochloric Acid SCHEMBL11197387 0.82 PRKCI (0.45) HTR2AKDM4EALDH1A1HTR2CKHK
SCHEMBL11204218 0.82 KDM4E (0.41) HTR2AKDM4EALDH1A1HTR2CHRH1
Hydrochloric Acid SCHEMBL11198496 0.81 KDM4E (0.40) HTR2AKDM4EALDH1A1HTR2CHRH1
SCHEMBL11197339 0.81 HTR2C (0.39) HTR2AKDM4EALDH1A1HTR2CKHK
SCHEMBL11203370 0.79 IKBKB (0.40) HTR2AKDM4EALDH1A1HTR2CKHK
SCHEMBL11205242 0.77 MAPT (0.45) KDM4EALDH1A1SMN1; SMN2CASP1TSHR
SCHEMBL11200202 0.77 KHK (0.38) HTR2AKDM4EALDH1A1HTR2CKHK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0082023-A2 Thienopyrimidine derivatives, their preparation and their medical use SANKYO COMPANY LIMITED (JP) 1983-06-22 EP disclosed