SCHEMBL11201445

SCHEMBL11201445

CC(C)c1csc2nc(N3CCNCC3)nc(NCCO)c12

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.41
SYK P43405 1/20 0.38
KHK P50053 2/20 0.37
CCNE1 P24864 2/20 0.36
CDK2 P24941 2/20 0.36
HRH4 Q9H3N8 2/20 0.36
HTR2A P28223 1/20 0.36
HTR3A P46098 1/20 0.36
ALDH1A1 P00352 3/20 0.35
GLA P06280 1/20 0.35
KDM4E B2RXH2 3/20 0.35
HTR2C P28335 1/20 0.35
ALOX15 P16050 2/20 0.35
USP2 O75604 1/20 0.35
LMNA P02545 1/20 0.35
ELANE P08246 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11197538 0.86 PRKCI (0.41) ESR1SYKKHKHRH4HTR3A
SCHEMBL11201137 0.85 ESR1 (0.39) ESR1HRH4HTR2AHTR3AALDH1A1
SCHEMBL11206366 0.84 HTR2A (0.39) ESR1KHKHRH4HTR2AALDH1A1
SCHEMBL11200579 0.84 SYK (0.40) ESR1SYKKHKCCNE1CDK2
Hydrochloric Acid SCHEMBL11202845 0.83 HTR2A (0.39) ESR1KHKHRH4HTR2AALDH1A1
SCHEMBL11202898 0.79 ELANE (0.35) ESR1KHKHRH4HTR2AHTR2C
SCHEMBL11204218 0.77 KDM4E (0.41) HTR2AALDH1A1KDM4EHTR2CUSP2
Hydrochloric Acid SCHEMBL11198496 0.76 KDM4E (0.40) HTR2AALDH1A1KDM4EHTR2CUSP2
SCHEMBL11201871 0.75 PRKCI (0.41) ESR1KHKHTR2AHTR2C
SCHEMBL11205170 0.74 ALDH1A1 (0.42) SYKKHKHRH4HTR3AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0082023-A2 Thienopyrimidine derivatives, their preparation and their medical use SANKYO COMPANY LIMITED (JP) 1983-06-22 EP disclosed