SCHEMBL11207797

SCHEMBL11207797

Cc1cc(N)c(N)cc1[N+](=O)[O-]

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 7/20 0.59
CYP3A4 P08684 5/20 0.59
ALDH1A1 P00352 3/20 0.59
RECQL P46063 1/20 0.59
TDP1 Q9NUW8 5/20 0.50
GAA P10253 1/20 0.50
MAPT P10636 2/20 0.47
MEN1 O00255 1/20 0.47
POLB P06746 1/20 0.47
KMT2A Q03164 1/20 0.47
ALOX15 P16050 1/20 0.47
HSD17B10 Q99714 1/20 0.45
CYP1A2 P05177 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30578482 1.00 TSHR (0.59) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL11219818 0.91 TSHR (0.59) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL30578459 0.91 TSHR (0.59) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL7461987 0.89 TSHR (0.57) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL1464001 0.89 TSHR (0.57) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL30675090 0.89 TSHR (0.57) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL6672279 0.89 TSHR (0.57) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL9652342 0.84 TSHR (0.57) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL2988066 0.84 TSHR (0.52) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL9464332 0.84 ALDH1A1 (0.62) TSHRCYP3A4ALDH1A1RECQLTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020155925-A1 NITROALKYL QUINOXALINE OR DERIVATIVE THEREOF, AMINOALKYL QUINOXALINE OR DERIVATIVE THEREOF, AND SYNTHESIS METHOD THEREFOR 上海交通大学 2020-08-06 WO claimed
CN-109608406-A A kind of nitro alkyl quinoxaline or derivatives thereof, aminoalkyl quinoxaline or derivatives thereof and its synthetic method 上海交通大学 2019-04-12 CN claimed
CN-108840827-A The method of the quinoxaline that one-step synthesis method dinitro replaces or derivatives thereof 同济大学 2018-11-20 CN claimed
WO-2020155925-A1 NITROALKYL QUINOXALINE OR DERIVATIVE THEREOF, AMINOALKYL QUINOXALINE OR DERIVATIVE THEREOF, AND SYNTHESIS METHOD THEREFOR 上海交通大学 2020-08-06 WO disclosed
CN-109608406-A A kind of nitro alkyl quinoxaline or derivatives thereof, aminoalkyl quinoxaline or derivatives thereof and its synthetic method 上海交通大学 2019-04-12 CN disclosed
CN-108840827-A The method of the quinoxaline that one-step synthesis method dinitro replaces or derivatives thereof 同济大学 2018-11-20 CN disclosed
EP-0012909-B1 BENZIMIDAZOLYL-2-ALKANE-PHOSPHONIC ACIDS AND THEIR SALTS, PROCESS FOR THEIR PREPARATION AND THEIR USE AS CORROSION INHIBITORS OR WETTING AGENTS BAYER AG (DE) 1983-06-15 EP disclosed
US-4278791-A CORROSION RESISTANCE, WETTING AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1981-07-14 US disclosed
EP-0001246-B1 PREPARATION OF 2-(3'- OR 4'-AMINOPHENYL)-5(OR 6)-AMINOBENZIMIDAZOLES CASSELLA Aktiengesellschaft (DE) 1981-02-25 EP disclosed
EP-0012909-A1 Benzimidazolyl-2-alkane-phosphonic acids and their salts, process for their preparation and their use as corrosion inhibitors or wetting agents BAYER AG (DE) 1980-07-09 EP disclosed
US-4192947-A REACTING DIAMINO NITROBENZENE WITH NITROBENZOYL CHLORIDE, CYCLIZING ANILIDE IN AQUEOUS ALKALI, REDUCING NITRO GROUPS WITH SULFIDE CASSELLA AKTIENGESELLSCHAFT (DE) 1980-03-11 US disclosed
EP-0001246-A1 Preparation of 2-(3'- or 4'-aminophenyl)-5(or 6)-aminobenzimidazoles CASSELLA Aktiengesellschaft (DE) 1979-04-04 EP disclosed
US-4138568-A NITRO-O-PHENYLENEDIAMINE, UREA, HALOBENZENE SOLVENT CIBA-GEIGY CORPORATION (US) 1979-02-06 US disclosed