Imidazole

Imidazole

SCHEMBL11208968

O=C(O)[C@@H](Cc1c[nH]cn1)NCc1ccccc1.c1c[nH]cn1

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPR142 Q7Z601 7/20 0.38
ALDH1A1 P00352 3/20 0.35
KDM4A O75164 1/20 0.35
KDM4B O94953 1/20 0.35
KDM5C P41229 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
POLB P06746 1/20 0.34
CYP3A4 P08684 1/20 0.34
AGTR2 P50052 1/20 0.34
RAB9A P51151 1/20 0.33
PSMB5 P28074 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Imidazole SCHEMBL27561511 1.00 GPR142 (0.38) GPR142ALDH1A1KDM4AKDM4BKDM5C
Imidazole SCHEMBL9152956 1.00 GPR142 (0.38) GPR142ALDH1A1KDM4AKDM4BKDM5C
Imidazole SCHEMBL27609343 0.99 GPR142 (0.38) GPR142ALDH1A1KDM4AKDM4BKDM5C
SCHEMBL466341 0.91 GAA (0.40) GPR142ALDH1A1GAAMAPTPOLB
SCHEMBL1643961 0.91 GAA (0.40) GPR142ALDH1A1GAAMAPTPOLB
SCHEMBL466340 0.91 GAA (0.40) GPR142ALDH1A1GAAMAPTPOLB
Imidazole SCHEMBL27889109 0.88 GPR142 (0.39) GPR142RAB9A
Imidazole SCHEMBL7422560 0.81 NR1H4 (0.37) GPR142RAB9A
SCHEMBL6384640 0.81 MC5R (0.39) GPR142
SCHEMBL6447871 0.79 SIRT2 (0.48) ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0021620-B1 WATER-SOLUBLE PEPTIDES AFFECTING GONADAL FUNCTION THE SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 1983-02-23 EP disclosed
US-4244946-A LUTEINIZING-HORMONE RELEASING FACTOR AGONISTS AS ANTIFERTILITY AGENTS THE SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 1981-01-13 US disclosed
EP-0021620-A1 Water-soluble peptides affecting gonadal function THE SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 1981-01-07 EP disclosed