SCHEMBL11209604

SCHEMBL11209604

CCCCC1CCc2cc(C(=O)Oc3ccc(C#N)cc3)ccc2C1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.46
MGLL Q99685 2/20 0.42
CYP3A4 P08684 2/20 0.41
CYP2C8 P10632 2/20 0.41
S1PR3 Q99500 2/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
SGPL1 O95470 2/20 0.40
CYP19A1 P11511 2/20 0.40
PPARD Q03181 1/20 0.38
PPARA Q07869 1/20 0.38
PRSS1 P07477 1/20 0.38
ACR P10323 1/20 0.38
S1PR1 P21453 3/20 0.38
SRD5A1 P18405 1/20 0.38
SRD5A2 P31213 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11075730 0.97 MCHR1 (0.46) MCHR1MGLLCYP3A4CYP2C8S1PR3
SCHEMBL11209612 0.96 CYP3A4 (0.46) MCHR1MGLLCYP3A4CYP2C8S1PR3
SCHEMBL11211358 0.96 CYP3A4 (0.46) MCHR1MGLLCYP3A4CYP2C8S1PR3
SCHEMBL11209532 0.96 CYP3A4 (0.46) MCHR1MGLLCYP3A4CYP2C8S1PR3
SCHEMBL11214851 0.94 MCHR1 (0.48) MCHR1MGLLCYP3A4CYP2C8S1PR3
SCHEMBL11209164 0.90 MCHR1 (0.49) MCHR1MGLLCYP19A1PPARDPPARA
SCHEMBL11206793 0.86 MCHR1 (0.48) MCHR1CYP3A4CYP2C8S1PR3CYP2D6
SCHEMBL14525798 0.85 MCHR1 (0.42) MCHR1CYP3A4CYP2C8S1PR3CYP2D6
SCHEMBL11213381 0.85 MCHR1 (0.47) MCHR1CYP3A4CYP2C8S1PR3CYP2D6
SCHEMBL11207970 0.85 CYP3A4 (0.48) MCHR1CYP3A4CYP2C8S1PR3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4391731-A Hydrogenated naphthalenes HOFFMANN-LA ROCHE INC. (US) 1983-07-05 US disclosed
EP-0047817-A2 Hydrogenated naphthalines, their preparation and application, and mixtures containing such naphthalines F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1982-03-24 EP disclosed