SCHEMBL11210049

SCHEMBL11210049

CC(=O)n1c(=O)sc2c(Cl)cccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 5/20 0.45
POLB P06746 1/20 0.42
MAPT P10636 3/20 0.38
TSHR P16473 1/20 0.38
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
NPSR1 Q6W5P4 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4617255 0.77 MEN1 (0.38) NOTUMMAPTTSHRHDAC3HDAC4
SCHEMBL4616310 0.74 POLB (0.50) POLBMAPTTSHRNPSR1ALDH1A1
SCHEMBL9806019 0.73 ASAH1 (0.47) POLBMAPTNPSR1CYP1A2CYP3A4
SCHEMBL9806051 0.72 HTT (0.48) TSHRNPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL22045678 0.66 PARP1 (0.36) NOTUMPOLBHDAC3HDAC4HDAC1
SCHEMBL3314327 0.64 POLB (0.61) NOTUMPOLBMAPTTSHRNPSR1
SCHEMBL11397522 0.63 PARP10 (0.46) NOTUMPOLBTSHRHDAC3HDAC4
SCHEMBL5277846 0.63 MAPT (0.40) NOTUMMAPTCYP1A2CYP3A4CYP2C19
SCHEMBL17621007 0.62 KDM4E (0.37) TSHRHDAC3HDAC4HDAC1HDAC7
SCHEMBL11649328 0.61 PTGS2 (0.35) POLBMAPTTSHRHDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0039440-B1 MEDICINES CONTAINING SUBSTITUTED BENZOTHIAZOL-2-(3H)-ONES Dr. Karl Thomae GmbH (DE) 1983-06-22 EP disclosed
US-4353919-A Analgesic and antipyretic pharmaceutical compositions containing a benzothiazol-2(3H)-one DR. KARL THOMAE GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1982-10-12 US disclosed
EP-0039440-A1 Medicines containing substituted benzothiazol-2-(3H)-ones Dr. Karl Thomae GmbH (DE) 1981-11-11 EP disclosed