SCHEMBL11210180

SCHEMBL11210180

CSC(C#N)c1cccc(Oc2ccccc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
CYP2D6 P10635 1/20 0.48
ALOX5 P09917 2/20 0.46
ALDH1A1 P00352 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
AKR1C3 P42330 1/20 0.40
MAOB P27338 1/20 0.40
TSHR P16473 2/20 0.38
LTA4H P09960 1/20 0.38
SGMS2 Q8NHU3 1/20 0.37
FAAH O00519 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
HTT P42858 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9049616 0.84 PTGS1 (0.53) PTGS1MEN1KMT2ACYP2D6ALOX5
SCHEMBL11211316 0.80 PTGS1 (0.43) PTGS1MEN1KMT2ACYP2D6ALOX5
SCHEMBL9493266 0.79 TSHR (0.46) MEN1KMT2AALDH1A1AKR1C3TSHR
SCHEMBL7035268 0.79 PTGS1 (0.57) PTGS1MEN1KMT2ACYP2D6ALOX5
SCHEMBL31542598 0.79 PTGS1 (0.57) PTGS1MEN1KMT2ACYP2D6ALOX5
SCHEMBL24106552 0.79 PTGS1 (0.57) PTGS1MEN1KMT2ACYP2D6ALOX5
SCHEMBL15978566 0.79 PTGS1 (0.57) PTGS1MEN1KMT2ACYP2D6ALOX5
SCHEMBL9664012 0.78 ALOX5 (0.55) PTGS1MEN1KMT2ACYP2D6ALOX5
SCHEMBL4449688 0.77 PTGS1 (0.50) PTGS1MEN1KMT2ACYP2D6ALOX5
SCHEMBL13886757 0.77 PTGS1 (0.50) PTGS1MEN1KMT2ACYP2D6ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0025262-B1 ALPHA-THIO-ALPHA-ARYL-SUBSTITUTED ALKANONITRILES, PROCESS FOR THEIR PREPARATION, PROCESS FOR PREPARING ALPHA-ARYL-SUBSTITUTED ALKANONITRILES AND THE CORRESPONDING CARBOXYLIC ACIDS THEREFROM AND PROCESS FOR PREPARING INTERMEDIATES SAGAMI CHEMICAL RESEARCH CENTER (JP) 1983-10-05 EP disclosed
US-4340740-A Alpha-thio-alpha-aryl-substituted alkanonitrile and process for preparing alpha-aryl-substituted alkanonitrile therefrom SAGAMI CHEMICAL RESEARCH CENTER (JP) 1982-07-20 US disclosed
EP-0025262-A2 Alpha-thio-alpha-aryl-substituted alkanonitriles, process for their preparation, process for preparing alpha-aryl-substituted alkanonitriles and the corresponding carboxylic acids therefrom and process for preparing intermediates SAGAMI CHEMICAL RESEARCH CENTER (JP) 1981-03-18 EP disclosed