SCHEMBL11212944

SCHEMBL11212944

CC(=O)O[C@@H]1C[C@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1NCC(=O)C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SHBG P04278 5/20 0.52
CYP3A4 P08684 10/20 0.51
LMNA P02545 8/20 0.51
ALDH1A1 P00352 7/20 0.51
MAPT P10636 6/20 0.51
SMN1; SMN2 Q16637 5/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
TSHR P16473 5/20 0.50
MAPK1 P28482 4/20 0.50
NR3C1 P04150 4/20 0.50
PGR P06401 4/20 0.50
AR P10275 4/20 0.50
SERPINA6 P08185 4/20 0.50
CYP2C9 P11712 3/20 0.50
GPBAR1 Q8TDU6 3/20 0.50
SIGMAR1 Q99720 3/20 0.50
CYP2C19 P33261 2/20 0.50
HIF1A Q16665 2/20 0.50
NR1I2 O75469 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11209590 0.87 SHBG (0.64) SHBGCYP3A4LMNAALDH1A1MAPT
SCHEMBL11212061 0.84 CYP19A1 (0.48) CYP3A4LMNAMAPTKMT2ACYP19A1
SCHEMBL11212950 0.80 SHBG (0.53) SHBGCYP3A4LMNAALDH1A1MAPT
SCHEMBL11228601 0.76 SHBG (0.58) SHBGCYP3A4LMNAALDH1A1MAPT
SCHEMBL2600420 0.73 CYP3A4 (0.79) SHBGCYP3A4LMNAALDH1A1MAPT
SCHEMBL18438757 0.73 CYP3A4 (0.79) SHBGCYP3A4LMNAALDH1A1MAPT
SCHEMBL15369348 0.73 CYP3A4 (0.79) SHBGCYP3A4LMNAALDH1A1MAPT
SCHEMBL7996078 0.73 CYP3A4 (0.79) SHBGCYP3A4LMNAALDH1A1MAPT
SCHEMBL2082800 0.73 CYP3A4 (0.79) SHBGCYP3A4LMNAALDH1A1MAPT
SCHEMBL4617560 0.73 CYP3A4 (0.79) SHBGCYP3A4LMNAALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0033561-B1 NOVEL 17-AMINO-16-HYDROXY STEROIDS OF THE ANDROSTANE AND OESTRANE SERIES AND DERIVATIVES THEREOF, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS AKZO N.V. (NL) 1983-05-11 EP disclosed
US-4330539-A Novel 17-amino-16-hydroxy steroids of the androstane and oestrane series and derivatives thereof AKZO NV (NL) 1982-05-18 US disclosed
EP-0033561-A1 Novel 17-amino-16-hydroxy steroids of the androstane and oestrane series and derivatives thereof, processes for their preparation and pharmaceutical compositions AKZO N.V. (NL) 1981-08-12 EP disclosed