SCHEMBL11213809

SCHEMBL11213809

NC(C=O)c1ccc2[nH]c(=O)oc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 4/20 0.50
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
OGT O15294 1/20 0.43
CREBBP Q92793 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
KMO O15229 1/20 0.41
NOS3 P29474 3/20 0.39
NOS2 P35228 3/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
ADRA2A P08913 1/20 0.39
TSHR P16473 1/20 0.39
THPO P40225 1/20 0.39
BLM P54132 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ALPL P05186 2/20 0.39
SMYD3 Q9H7B4 2/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9278834 0.86 NOS1 (0.49) NOS1PDE3BPDE3AOGTCREBBP
SCHEMBL13080918 0.81 NOS1 (0.46) NOS1PDE3BPDE3AOGTCREBBP
SCHEMBL9909873 0.77 NOS1 (0.61) NOS1PDE3BPDE3AOGTCREBBP
SCHEMBL2547913 0.74 NOS1 (0.57) NOS1PDE3BPDE3AOGTCREBBP
SCHEMBL18713322 0.73 NOS1 (0.56) NOS1PDE3BPDE3AOGTCREBBP
Hydrochloric Acid SCHEMBL10538242 0.73 NOS1 (0.47) NOS1PDE3BPDE3AOGTCREBBP
SCHEMBL18552760 0.72 NOS1 (0.54) NOS1PDE3BPDE3AOGTCREBBP
SCHEMBL13969518 0.72 NOS1 (0.54) NOS1PDE3BPDE3AOGTCREBBP
SCHEMBL3600957 0.71 NOS1 (0.58) NOS1PDE3BPDE3AOGTCREBBP
SCHEMBL22382321 0.71 NOS1 (0.49) NOS1PDE3BPDE3AOGTCREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1982001186-A1 NOVEL BENZOXAZOLINONES,SUBSTITUTED IN THE 6-POSITION BY AN AMINOALCOHOL CHAIN OR AMINO-KETONE CHAIN,THEIR PREPARATION AND THEIR USE IN PHARMACEUTICAL PREPARATIONS BUSCH N 1982-04-15 WO disclosed