SCHEMBL11221097

SCHEMBL11221097

C=CCOC(=O)CCc1cccnc1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 9/20 0.49
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
PKM P14618 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CASP1 P29466 1/20 0.45
NAPRT Q6XQN6 1/20 0.44
CHRNA7 P36544 2/20 0.43
TRPV1 Q8NER1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9280186 0.85 NAPRT (0.54) TBXAS1KDM4ELMNATDP1CYP1A2
SCHEMBL250955 0.82 TDP1 (0.68) ALDH1A1TDP1CYP3A4PKMSMN1; SMN2
SCHEMBL3957320 0.81 CYP4F2 (0.55) TBXAS1ALDH1A1TDP1
SCHEMBL31556473 0.80 TBXAS1 (0.58) TBXAS1KDM4EALDH1A1LMNACYP1A2
Hydrochloric Acid SCHEMBL18230734 0.79 CYP4F2 (0.54) TBXAS1ALDH1A1TDP1
SCHEMBL304802 0.79 TDP1 (0.60) TBXAS1KDM4EALDH1A1LMNATDP1
Hydrochloric Acid SCHEMBL27552763 0.79 CYP4F2 (0.54) TBXAS1ALDH1A1TDP1
SCHEMBL10663309 0.79 TSHR (0.45) KDM4EALDH1A1TDP1CYP3A4PKM
SCHEMBL8476744 0.77 TBXAS1 (0.55) TBXAS1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL64891 0.77 TBXAS1 (0.59) TBXAS1KDM4EALDH1A1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0070185-A1 Preparation of lower alkyl 2-formyl-3-(6-methyl-3-pyridinyl)-propionates SMITHKLINE BECKMAN CORPORATION (US) 1983-01-19 EP claimed
EP-0070185-A1 Preparation of lower alkyl 2-formyl-3-(6-methyl-3-pyridinyl)-propionates SMITHKLINE BECKMAN CORPORATION (US) 1983-01-19 EP disclosed
EP-0070185-A1 Preparation of lower alkyl 2-formyl-3-(6-methyl-3-pyridinyl)-propionates SMITHKLINE BECKMAN CORPORATION (US) 1983-01-19 EP disclosed
US-4153795-A Cobalt pyridyl catalysts for hydroformylation DIRECTOR-GENERAL OF THE AGENCY OF INDUSTRIAL SCIENCE AND TECHNOLOGY (JP) 1979-05-08 US disclosed