SCHEMBL11223955

SCHEMBL11223955

COc1cc2c(cc1OC)C(CCCCCl)(c1ccc(F)cc1)OCC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 4/20 0.41
BCHE P06276 1/20 0.38
SLC6A2 P23975 2/20 0.37
HTR2C P28335 2/20 0.37
ADRA1A P35348 2/20 0.37
HRH1 P35367 2/20 0.37
OPRM1 P35372 2/20 0.37
DRD3 P35462 2/20 0.37
HTR2B P41595 2/20 0.37
KCNH2 Q12809 2/20 0.37
NPC1 O15118 1/20 0.37
SLC22A1 O15245 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CHRM2 P08172 1/20 0.37
HTR1A P08908 1/20 0.37
CHRM1 P11229 1/20 0.37
DRD1 P21728 1/20 0.37
ACHE P22303 1/20 0.37
HRH2 P25021 1/20 0.37
ADRA1D P25100 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11224396 0.97 SLC6A4 (0.41) SLC6A4BCHESLC6A2HTR2CADRA1A
SCHEMBL11220962 0.95 SLC6A4 (0.40) SLC6A4BCHESLC6A2HTR2CADRA1A
SCHEMBL11225546 0.91 SLC6A4 (0.41) SLC6A4BCHESLC6A2HTR2CADRA1A
SCHEMBL11222322 0.88 SLC6A4 (0.40) SLC6A4BCHESLC6A2HTR2CADRA1A
SCHEMBL11668322 0.86 SLC6A4 (0.57) SLC6A4SLC6A2HTR2CADRA1AHRH1
SCHEMBL11419267 0.85 HTR1A (0.36) SLC6A4ADRA1ADRD3HTR1AADRA1D
SCHEMBL11536230 0.84 KMT2A (0.36) SLC6A4BCHE
SCHEMBL11668436 0.83 KMT2A (0.39) SLC6A4ALDH1A1CYP2D6
SCHEMBL11221675 0.83 SLC6A4 (0.39) SLC6A4BCHESLC6A2HTR2CADRA1A
SCHEMBL9134820 0.80 KDM4E (0.45) HTR2CALDH1A1HTR1AHTR2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4352805-A BENZOXEPINE DERIVATIVES THE UPJOHN COMPANY (US) 1982-10-05 US disclosed
US-4312868-A HYPOTENSIVE, ANTIPSYCHOTIC THE UPJOHN COMPANY (US) 1982-01-26 US disclosed
US-4251526-A HYPOTENSIVE AGENTS AND ANTIPSYCHOTIC PHARMACIA & UPJOHN COMPANY 1981-02-17 US disclosed
US-4250181-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-02-10 US disclosed
US-4250175-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS PHARMACIA & UPJOHN COMPANY 1981-02-10 US disclosed
US-4247553-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-01-27 US disclosed
US-4179510-A ISOCHROMANS AND 2-BENZOXEPINS THE UPJOHN COMPANY (US) 1979-12-18 US disclosed
US-4153612-A 2-Benzoxepins THE UPJOHN COMPANY (US) 1979-05-08 US disclosed