SCHEMBL11224734

SCHEMBL11224734

CC(=O)/C=C(\C)Nc1cc(-c2cccnc2C)c[nH]c1=O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITK Q08881 7/20 0.42
TTK P33981 3/20 0.41
AURKB Q96GD4 2/20 0.41
INCENP Q9NQS7 2/20 0.41
AURKA O14965 1/20 0.41
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
GPR142 Q7Z601 6/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
KIT P10721 2/20 0.38
SRC P12931 2/20 0.38
FLT3 P36888 2/20 0.38
KDR P35968 1/20 0.38
ABL1 P00519 1/20 0.36
TDO2 P48775 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11224738 1.00 ITK (0.42) ITKTTKAURKBINCENPAURKA
SCHEMBL11228274 0.82 MKNK1 (0.39) ITKTTKAURKBINCENPAURKA
SCHEMBL11228272 0.82 MKNK1 (0.39) ITKTTKAURKBINCENPAURKA
SCHEMBL11234332 0.80 TTK (0.51) ITKTTKAURKBINCENPAURKA
SCHEMBL11234330 0.80 TTK (0.51) ITKTTKAURKBINCENPAURKA
SCHEMBL11219801 0.79 ITK (0.61) ITKTTKAURKBINCENPAURKA
SCHEMBL11219799 0.79 ITK (0.61) ITKTTKAURKBINCENPAURKA
SCHEMBL11228315 0.76 ITK (0.44) ITKTTKAURKBINCENPAURKA
SCHEMBL11228318 0.76 ITK (0.44) ITKTTKAURKBINCENPAURKA
SCHEMBL11231633 0.76 CCNC (0.48) ITKTTKAURKBINCENPAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4362735-A 3-[(3-Oxo-1-butenyl)amino]-5-(pyridinyl)-2(1H)-pyridinones and their cardiotonic use STERLING DRUG INC. (US) 1982-12-07 US disclosed