SCHEMBL11225236

SCHEMBL11225236

C[C@H](NC(=O)[C@H](C)NP(=O)(O)O)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.46
MME P08473 5/20 0.43
CPA1 P15085 1/20 0.43
ACE2 Q9BYF1 1/20 0.43
LTA4H P09960 3/20 0.36
ANPEP P15144 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
MMP1 P03956 1/20 0.35
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
MMP8 P22894 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL72229 0.84 ACE (0.48) ACELTA4HCA12CA1CA2
SCHEMBL72230 0.84 ACE (0.48) ACELTA4HCA12CA1CA2
SCHEMBL18098146 0.73 MME (0.48) ACEMMECPA1ACE2LTA4H
SCHEMBL21375005 0.73 ACE (0.59) ACEMMECPA1ACE2
SCHEMBL6468859 0.73 ACE (0.59) ACEMMECPA1ACE2
SCHEMBL23142762 0.73 MME (0.48) ACEMMECPA1ACE2LTA4H
SCHEMBL15307782 0.73 MME (0.48) ACEMMECPA1ACE2LTA4H
SCHEMBL13598642 0.73 MME (0.48) ACEMMECPA1ACE2LTA4H
SCHEMBL13165106 0.73 MME (0.48) ACEMMECPA1ACE2LTA4H
SCHEMBL15080628 0.73 MME (0.48) ACEMMECPA1ACE2LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4316896-A Aminoacid derivatives as antihypertensives MERCK & CO., INC. (US) 1982-02-23 US disclosed
EP-0009183-B1 PHOSPHORYL AMINOACID DERIVATIVES AND COMPOSITION FOR TREATING HYPERTENSION CONTAINING THE SAME MERCK & CO. INC. (US) 1981-10-21 EP disclosed
EP-0009183-A1 Phosphoryl aminoacid derivatives and composition for treating hypertension containing the same MERCK & CO. INC. (US) 1980-04-02 EP disclosed