SCHEMBL11230795

SCHEMBL11230795

CCOC(=O)CS(=O)(=O)c1ccc(CC)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.73
GAA P10253 3/20 0.60
HSD11B1 P28845 1/20 0.50
PHGDH O43175 1/20 0.47
CA2 P00918 2/20 0.47
CA9 Q16790 2/20 0.47
LMNA P02545 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
NPSR1 Q6W5P4 1/20 0.46
ALDH1A1 P00352 4/20 0.45
HCRTR2 O43614 1/20 0.44
CA12 O43570 1/20 0.44
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CYP4F2 P78329 1/20 0.42
CYP4A11 Q02928 1/20 0.42
KDM4E B2RXH2 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MEN1 O00255 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27272113 0.87 KMT2A (0.69) KMT2AGAAHSD11B1PHGDHCA2
SCHEMBL2178479 0.86 KMT2A (0.78) KMT2AGAAHSD11B1CA2CA9
SCHEMBL23049758 0.86 KMT2A (0.68) KMT2AGAAHSD11B1PHGDHCA2
SCHEMBL23049909 0.86 KMT2A (0.55) KMT2AGAAHSD11B1PHGDHCA2
SCHEMBL18503840 0.85 KMT2A (1.00) KMT2AGAAHSD11B1PHGDHCA2
SCHEMBL23049753 0.85 KMT2A (0.53) KMT2AGAAPHGDHCA2ALDH1A1
SCHEMBL23049646 0.84 KMT2A (0.54) KMT2AGAAPHGDHCA2CA9
SCHEMBL23049630 0.84 KMT2A (0.54) KMT2AGAAPHGDHCA2CA9
SCHEMBL23049717 0.84 KMT2A (0.54) KMT2AGAAHSD11B1PHGDHCA2
SCHEMBL23703133 0.83 KMT2A (0.73) KMT2AGAAHSD11B1PHGDHCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1018548-B CARBOXYLIC ACID DERIVATIVES, PROCESSES FOR PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1992-10-07 CN claimed
EP-3596064-B1 TOSYLACETATE BASED COMPOUNDS AND DERIVATIVES THEREOF AS PHGDH INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2021-03-03 EP disclosed
US-4326066-A Triazolyl coumarin compounds, processes for their preparation and their use as whiteners and laser dyestuffs BAYER AKTIENGESELLSCHAFT (DE) 1982-04-20 US disclosed