SCHEMBL2178479

SCHEMBL2178479

CCOC(=O)CS(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.78

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.78
GAA P10253 3/20 0.63
ALDH1A1 P00352 5/20 0.61
CA2 P00918 1/20 0.56
CA9 Q16790 1/20 0.56
RECQL P46063 1/20 0.54
HSD11B1 P28845 2/20 0.52
MAPT P10636 1/20 0.50
HSD17B10 Q99714 1/20 0.50
LMNA P02545 2/20 0.49
NPSR1 Q6W5P4 1/20 0.49
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
PKM P14618 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13299621 0.95 KMT2A (0.71) KMT2AGAAALDH1A1CA2CA9
SCHEMBL18503840 0.88 KMT2A (1.00) KMT2AGAAALDH1A1CA2CA9
SCHEMBL1939652 0.86 KMT2A (0.73) KMT2AGAAALDH1A1CA2CA9
SCHEMBL11230795 0.86 KMT2A (0.73) KMT2AGAAALDH1A1CA2CA9
SCHEMBL23703133 0.86 KMT2A (0.73) KMT2AGAAALDH1A1CA2CA9
SCHEMBL25061922 0.86 KMT2A (0.73) KMT2AGAAALDH1A1HSD11B1MAPT
SCHEMBL1464359 0.86 KMT2A (0.73) KMT2AGAAALDH1A1HSD11B1NPSR1
SCHEMBL2024141 0.86 KMT2A (0.73) KMT2AGAAALDH1A1CA9RECQL
SCHEMBL5860960 0.85 KMT2A (0.71) KMT2AGAAALDH1A1HSD11B1MAPT
SCHEMBL8249922 0.85 KMT2A (0.71) KMT2AGAAALDH1A1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 58 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230348450-A1 CARBOXYLIC ACID-CONTAINING COMPOUNDS AS MODULATORS OF BIS-PHOSPHOGLYCERATE MUTASE FOR THE TREATMENT OF SICKLE CELL DISEASE GENZYME CORPORATION 2023-11-02 US disclosed
US-20230321016-A1 COMBINATION THERAPY FOR TREATING CANCER GONGWIN BIOPHARM CO., LTD (TW) 2023-10-12 US disclosed
US-11752118-B2 Method for treating melanoma GONGWIN BIOPHARM CO., LTD (TW) 2023-09-12 US disclosed
US-11752160-B2 Method for reducing fat by administering benzenesulfonamide compositions GONGWIN BIOPHARM CO., LTD (TW) 2023-09-12 US disclosed
US-20230054928-A1 METHOD FOR PREPARING CARBONYL SULFONE SOOCHOW UNIVERSITY (CN) 2023-02-23 US disclosed
US-10905769-B2 Peptide and peptide mimetic binding antagonists of polo-like kinase 1 polo box domain and methods of use THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH & HUMAN SERVICES (US) 2021-02-02 US disclosed
CN-111808003-A Preparation method of thioether 甘肃农业大学 2020-10-23 CN disclosed
CN-110054574-A A kind of synthetic method of fluorenylmethyloxycarbonyl -2,3- dehydrogenation-valine 上海吉奉生物科技有限公司 2019-07-26 CN disclosed
CN-102786373-B A kind of synthetic method of diazomethane compound SHENZHEN IPI BIOLOGICAL TECHNOLOGY CO., LTD. (CN) 2016-01-13 CN disclosed
CN-102786373-A Synthetic method of diazomethane compound SHENZHEN IPI BIOLOG TECHNOLOGY CO LTD 2012-11-21 CN disclosed
US-6342508-B1 ENZYME INHIBITORS FOR PROTECTION OF CONNECTIVE TISSUES AMERICAN CYANAMID COMPANY 2002-01-29 US disclosed
US-20020006922-A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors AMERICAN CYANAMID COMPANY (US) 2002-01-17 US disclosed
US-6331563-B1 LOW MOLECULAR WEIGHT, NON-PEPTIDE INHIBITORS OF MATRIX METALLOPROTEINASES AND TUMOR NECROSIS FACTOR-ALPHA CONVERTING ENZYME; TREATING ARTHRITIS, TUMOR METASTASIS, ABNORMAL WOUND HEALING, PERIODONTAL DISEASE, BONE DISEASE, INSULIN RESISTANCE WYETH HOLDINGS CORPORATION 2001-12-18 US disclosed
US-6288086-B1 COMPOUNDS SUCH AS 1-METHYL-4-(4-BUTOXY-BENZENESULFONYL) -PIPERIDINE-4-CARBOXYLIC ACID HYDROXYAMIDE USED TO TREAT ARTHRITIS, TUMOR METASTASIS, TISSUE ULCERATION, ABNORMAL WOUND HEALING, ETC.; LOW MOLECULAR WEIGHT AND NON-PEPTIDAL AMERICAN CYANAMID COMPANY 2001-09-11 US disclosed
US-6172057-B1 ANTIINFLAMMATORY AGENTS; ANTIARTHRITIC AGENTS; ANTITUMOR AGENTS AMERICAN CYANAMID COMPANY 2001-01-09 US disclosed
EP-1054858-A1 N-HYDROXY-2-(ALKYL, ARYL, OR HETEROARYL SULFANYL, SULFINYL OR SULFONYL)-3-SUBSTITUTED-ALKYL, ARYL OR HETEROARYLAMIDES AS MATRIX METALLOPROTEINASE INHIBITORS American Cyanamid Company (US) 2000-11-29 EP disclosed
WO-1999042436-A1 N-HYDROXY-2-(ALKYL, ARYL, OR HETEROARYL SULFANYL, SULFINYL OR SULFONYL)-3-SUBSTITUTED-ALKYL, ARYL OR HETEROARYLAMIDES AS MATRIX METALLOPROTEINASE INHIBITORS AMERICAN CYANAMID COMPANY (US) 1999-08-26 WO disclosed
US-5597776-A ANTAGONIST FOR HERBICIDES BASF AKTIENGESELLSCHAFT (DE) 1997-01-28 US disclosed
US-5145611-A Diabetes BOEHRINGER MANNHEIM GMBH (DE) 1992-09-08 US disclosed
US-4326066-A Triazolyl coumarin compounds, processes for their preparation and their use as whiteners and laser dyestuffs BAYER AKTIENGESELLSCHAFT (DE) 1982-04-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11752160-B2 Method for reducing fat by administering benzenesulfonamide compositions LIPE, FABP4, LIPA KMT2A 2032/4885GAA 128/4885ALDH1A1 728/4885
US-20230348450-A1 CARBOXYLIC ACID-CONTAINING COMPOUNDS AS MODULATORS OF BIS-PHOSPHOGLYCERATE MUTASE FOR THE TREATMENT OF SICKLE CELL DISEASE BPGM, PGAM1, PGM2 KMT2A 2181/4885GAA 9/4885ALDH1A1 326/4885
US-10905769-B2 Peptide and peptide mimetic binding antagonists of polo-like kinase 1 polo box domain and methods of use PLK1, POLR1E, POLK KMT2A 1885/4885GAA 2860/4885ALDH1A1 4834/4885
US-20230054928-A1 METHOD FOR PREPARING CARBONYL SULFONE TST, CBS, STS KMT2A 2093/4885GAA 707/4885ALDH1A1 297/4885
US-20230321016-A1 COMBINATION THERAPY FOR TREATING CANCER TP53, MCL1, TOP2B KMT2A 1380/4885GAA 1313/4885ALDH1A1 381/4885
US-11752118-B2 Method for treating melanoma TYR, MITF, BRAF KMT2A 1442/4885GAA 552/4885ALDH1A1 528/4885
US-20020006922-A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors MMP12, ADAM33, MMP2 KMT2A 3103/4885GAA 351/4885ALDH1A1 3024/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.