SCHEMBL11234892

SCHEMBL11234892

O=C(O)[C@]1(c2ccc(Sc3ccccc3)cc2)CCCN1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
AKR1C1 Q04828 1/20 0.37
EZH2 Q15910 1/20 0.36
MAOA P21397 2/20 0.36
MAOB P27338 2/20 0.36
ALOX5 P09917 1/20 0.32
ABL1 P00519 1/20 0.32
PTGIR P43119 1/20 0.32
RARB P10826 1/20 0.31
RARG P13631 1/20 0.31
RXRA P19793 1/20 0.31
RXRB P28702 1/20 0.31
RXRG P48443 1/20 0.31
BCL2 P10415 1/20 0.31
MCL1 Q07820 1/20 0.31
LTB4R Q15722 1/20 0.31
LTB4R2 Q9NPC1 1/20 0.31
SIRT1 Q96EB6 1/20 0.31
HTR2C P28335 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL435512 0.86 AKR1C1 (0.48) ALDH1A1AKR1C1HDAC4
SCHEMBL994596 0.86 AKR1C1 (0.48) ALDH1A1AKR1C1HDAC4
SCHEMBL10659448 0.86 AKR1C1 (0.48) ALDH1A1AKR1C1HDAC4
Hydrochloric Acid SCHEMBL8114403 0.84 AKR1C1 (0.47) ALDH1A1AKR1C1HDAC4
Hydrochloric Acid SCHEMBL8114401 0.84 AKR1C1 (0.47) ALDH1A1AKR1C1HDAC4
SCHEMBL11241224 0.83 AKR1C1 (0.40) ALDH1A1HPGDAKR1C1
Hydrochloric Acid SCHEMBL11247968 0.82 AKR1C1 (0.39) HPGDAKR1C1
SCHEMBL16057460 0.81 AKR1C1 (0.52) AKR1C1HDAC4
SCHEMBL11238790 0.80 SIRT1 (0.39) ALDH1A1HPGDAKR1C1SIRT1
SCHEMBL10483428 0.80 ESR2 (0.41) AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4316905-A HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1982-02-23 US disclosed