SCHEMBL11237600

SCHEMBL11237600

CC(=O)/C=C/Nc1cc(-c2ccncc2)c(C)[nH]c1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 12/20 0.51
PDE3A Q14432 12/20 0.51
AURKB Q96GD4 1/20 0.51
INCENP Q9NQS7 1/20 0.51
KDM4E B2RXH2 2/20 0.51
HPGD P15428 2/20 0.51
PDE4A P27815 2/20 0.51
PDE4B Q07343 2/20 0.51
PDE4C Q08493 2/20 0.51
PDE4D Q08499 2/20 0.51
PDE5A O76074 1/20 0.51
LMNA P02545 1/20 0.51
TSHR P16473 1/20 0.51
PTGS1 P23219 1/20 0.51
CYP2C19 P33261 1/20 0.51
BLM P54132 1/20 0.51
CCNC P24863 1/20 0.47
CDK8 P49336 1/20 0.47
CSNK1A1 P48729 1/20 0.38
CSNK1D P48730 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11237603 1.00 PDE3B (0.51) PDE3BPDE3AAURKBINCENPKDM4E
SCHEMBL11222392 0.85 PDE3B (0.54) PDE3BPDE3AAURKBINCENPKDM4E
SCHEMBL11222395 0.85 PDE3B (0.54) PDE3BPDE3AAURKBINCENPKDM4E
SCHEMBL11224300 0.84 PDE3B (0.57) PDE3BPDE3AAURKBINCENPKDM4E
SCHEMBL11224303 0.84 PDE3B (0.57) PDE3BPDE3AAURKBINCENPKDM4E
SCHEMBL11238639 0.81 PDE3B (0.57) PDE3BPDE3AAURKBINCENPKDM4E
SCHEMBL11232562 0.81 PDE3B (0.51) PDE3BPDE3AAURKBINCENPKDM4E
SCHEMBL11232554 0.81 PDE3B (0.51) PDE3BPDE3AAURKBINCENPKDM4E
SCHEMBL11222397 0.78 ITK (0.55) PDE3BPDE3AAURKBINCENPKDM4E
SCHEMBL11222394 0.78 ITK (0.55) PDE3BPDE3AAURKBINCENPKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4362735-A 3-[(3-Oxo-1-butenyl)amino]-5-(pyridinyl)-2(1H)-pyridinones and their cardiotonic use STERLING DRUG INC. (US) 1982-12-07 US disclosed