SCHEMBL11238008

SCHEMBL11238008

CCNc1ncc(-c2ccncc2)cc1C#N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 2/20 0.45
GSK3B P49841 2/20 0.45
PRKACA P17612 1/20 0.45
CDK8 P49336 1/20 0.45
CLK2 P49760 1/20 0.45
CDK9 P50750 1/20 0.45
CDK5 Q00535 1/20 0.45
PRKCQ Q04759 1/20 0.45
ROCK1 Q13464 1/20 0.45
DYRK1A Q13627 1/20 0.45
LRRK2 Q5S007 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
DYRK1B Q9Y463 1/20 0.45
PIK3CD O00329 2/20 0.42
PIK3CA P42336 2/20 0.42
PIK3CB P42338 2/20 0.42
CHEK1 O14757 1/20 0.42
LATS1 O95835 1/20 0.42
LATS2 Q9NRM7 1/20 0.42
PDE3B Q13370 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11247724 0.85 PIK3CD (0.44) GSK3AGSK3BPRKACACDK8CLK2
SCHEMBL7284439 0.85 PRKCH (0.46) GSK3AGSK3BPRKACACDK8CLK2
SCHEMBL7291065 0.85 ROCK1 (0.46) GSK3AGSK3BPRKACACDK8CLK2
SCHEMBL7284179 0.84 GLA (0.42) GSK3AGSK3BPRKACACDK8CLK2
SCHEMBL7292117 0.84 ROCK1 (0.43) GSK3AGSK3BPRKACACDK8CLK2
SCHEMBL7283041 0.83 CLK4 (0.39) GSK3AGSK3BPRKACACDK8CLK2
SCHEMBL6369146 0.83 KDM4E (0.42) GSK3AGSK3BPRKACACDK8CLK2
SCHEMBL7293503 0.82 PRKCD (0.48) GSK3AGSK3BPRKACACDK8CLK2
SCHEMBL4590900 0.82 KDM4E (0.55) GSK3AGSK3BCLK4ALDH1A1KDM4E
SCHEMBL7292623 0.81 PRKCD (0.44) GSK3AGSK3BPRKACACDK8CLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4362734-A 2-(Substituted-amino)-5-(pyridinyl-nicotinonitriles, and their cardiotonic use STERLING DRUG INC. (US) 1982-12-07 US disclosed