SCHEMBL11238385

SCHEMBL11238385

CC(=O)Nc1ccccc1C#CC1CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.43
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
KMT2A Q03164 3/20 0.41
KCNH2 Q12809 1/20 0.41
MEN1 O00255 1/20 0.41
HTT P42858 1/20 0.41
CREBBP Q92793 2/20 0.40
CYP1A2 P05177 2/20 0.40
GRM5 P41594 1/20 0.40
BRD4 O60885 1/20 0.40
LMNA P02545 1/20 0.39
CYP2C19 P33261 2/20 0.39
POLB P06746 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CETP P11597 1/20 0.38
HDAC3 O15379 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11222584 0.80 KCNH2 (0.46) TDP1ALDH1A1HPGDSMN1; SMN2KMT2A
SCHEMBL1464139 0.77 GRM5 (0.45) SMN1; SMN2KMT2AKCNH2MEN1HTT
SCHEMBL11240717 0.74 KCNH2 (0.41) TDP1ALDH1A1HPGDSMN1; SMN2KCNH2
SCHEMBL21430508 0.74 KDM4E (0.48) ALDH1A1HPGDSMN1; SMN2KMT2AKCNH2
SCHEMBL11232881 0.74 CREBBP (0.42) ALDH1A1HPGDKMT2AKCNH2CREBBP
SCHEMBL7515266 0.74 HSD17B10 (0.49) TDP1ALDH1A1HPGDSMN1; SMN2KMT2A
SCHEMBL28862901 0.73 CETP (0.42) ALDH1A1HPGDSMN1; SMN2BRD4LMNA
SCHEMBL10448319 0.72 ALDH1A1 (0.50) ALDH1A1HPGDSMN1; SMN2KMT2AHTT
SCHEMBL2231380 0.72 ALDH1A1 (0.63) ALDH1A1HPGDSMN1; SMN2KMT2AMEN1
SCHEMBL11230955 0.72 KCNH2 (0.50) TDP1ALDH1A1HPGDSMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4168320-A Ethynylbenzene compounds and derivatives thereof to treat inflammation, pain or fever WILLIAM H. RORER, INC. (US) 1979-09-18 US claimed
US-4365093-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1982-12-21 US disclosed
US-4296264-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1981-10-20 US disclosed
US-4288457-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1981-09-08 US disclosed
US-4264627-A Ethynylbenzene compounds and derivatives thereof to treat inflammation, pain or fever WILLIAM H. RORER, INC. (US) 1981-04-28 US disclosed
US-4171373-A Ethynylbenzene compounds and derivatives thereof to treat pain, fever and inflammation WILLIAM H. RORER, INC. (US) 1979-10-16 US disclosed
US-4168320-A Ethynylbenzene compounds and derivatives thereof to treat inflammation, pain or fever WILLIAM H. RORER, INC. (US) 1979-09-18 US disclosed
US-4166133-A ETHYNYLBENZENE COMPOUNDS AND DERIVATIVES THEREOF TO TREAT PAIN, FEVER AND INFLAMMATION WILLIAM H. RORER, INC. (US) 1979-08-28 US disclosed
US-4157449-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1979-06-05 US disclosed
US-4150148-A NITROSUBSTITUTED WILLIAM H. RORER, INC. (US) 1979-04-17 US disclosed
US-4120889-A Cyano ethynylbenzene compounds WILLIAM H. RORER, INC. (US) 1978-10-17 US disclosed
US-4120885-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1978-10-17 US disclosed
US-4105786-A ANTIINFLAMMATORY WILLIAM H. RORER, INC. (US) 1978-08-08 US disclosed
US-4101591-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1978-07-18 US disclosed
US-4096279-A Ethynylbenzene compounds and derivatives thereof in the treatment of pain fever and inflammation WILLIAM H. RORER, INC. (US) 1978-06-20 US disclosed
US-4094995-A ETHYNYLBENZENE COMPOUNDS AND DERIVATIVES THEREOF TO TREAT PAIN, FEVER AND INFLAMMATION WILLIAM H. RORER, INC. (US) 1978-06-13 US disclosed
US-4093737-A Ethynylbenzene compounds and derivatives thereof in the treatment of pain, fever or inflammation WILLIAM H. RORER, INC. (US) 1978-06-06 US disclosed
US-4075354-A ETHYNYLBENZENE COMPOUNDS AND DERIVATIVES THEREOF FOR TREATING PAIN FEVER AND INFLAMMATION WILLIAM H. RORER, INC. (US) 1978-02-21 US disclosed
US-3981932-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1976-09-21 US disclosed