SCHEMBL11239698

SCHEMBL11239698

CCC(=Cn1ccnc1)C(=O)c1ccc(Cl)cc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.50
CYP3A4 P08684 3/20 0.40
CYP19A1 P11511 2/20 0.39
ALDH1A1 P00352 6/20 0.39
POLB P06746 1/20 0.39
THRB P10828 1/20 0.39
RECQL P46063 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
HTT P42858 1/20 0.39
CYP1A2 P05177 1/20 0.38
GABRA1 P14867 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
ADRA2C P18825 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11239695 1.00 MAPT (0.50) MAPTCYP3A4CYP19A1ALDH1A1POLB
Hydrochloric Acid SCHEMBL11243888 0.99 MAPT (0.49) MAPTCYP3A4CYP19A1ALDH1A1POLB
Hydrochloric Acid SCHEMBL11243883 0.99 MAPT (0.49) MAPTCYP3A4CYP19A1ALDH1A1POLB
SCHEMBL11234000 0.84 MAPT (0.53) MAPTCYP3A4CYP19A1ALDH1A1MEN1
SCHEMBL11234002 0.84 MAPT (0.53) MAPTCYP3A4CYP19A1ALDH1A1MEN1
SCHEMBL11247102 0.83 MAPT (0.54) MAPTCYP3A4CYP19A1ALDH1A1TDP1
SCHEMBL11247103 0.83 MAPT (0.54) MAPTCYP3A4CYP19A1ALDH1A1TDP1
Hydrochloric Acid SCHEMBL10876102 0.81 MAPT (0.42) MAPTCYP3A4ALDH1A1TDP1LMNA
Hydrochloric Acid SCHEMBL10876112 0.81 MAPT (0.42) MAPTCYP3A4ALDH1A1TDP1LMNA
SCHEMBL10874271 0.79 MAPT (0.44) MAPTCYP3A4CYP19A1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4317831-A Antimicrobial derivatives of 3-(1H-imidazol-1-yl)-2-propen-1-ones E. R. SQUIBB & SONS, INC. (US) 1982-03-02 US disclosed
US-4273776-A Antibacterial and antifungal derivatives of 3-(1H-imidazol-1-yl)-2-propen-1-ones E. R. SQUIBB & SONS, INC. (US) 1981-06-16 US disclosed