SCHEMBL11240469

SCHEMBL11240469

COCCCNc1ncc(-c2ccncc2)cc1N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.51
TTK P33981 1/20 0.51
AURKB Q96GD4 1/20 0.51
INCENP Q9NQS7 1/20 0.51
LMNA P02545 2/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PDGFRB P09619 3/20 0.39
PDGFRA P16234 3/20 0.39
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
NTRK1 P04629 2/20 0.38
ALDH1A1 P00352 2/20 0.38
PRKCB P05771 1/20 0.38
PRKCA P17252 1/20 0.38
PRKCH P24723 1/20 0.38
PRKCE Q02156 1/20 0.38
PRKCQ Q04759 1/20 0.38
PRKCD Q05655 1/20 0.38
TLR7 Q9NYK1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11231162 0.84 LATS1 (0.49) AURKATTKAURKBINCENPLMNA
SCHEMBL11232478 0.83 PRKCD (0.51) AURKATTKAURKBINCENPPDGFRB
SCHEMBL11241274 0.82 GSK3B (0.46) AURKATTKAURKBINCENPHTT
SCHEMBL11227751 0.82 AURKA (0.45) AURKATTKAURKBINCENPROCK2
SCHEMBL11230984 0.80 POLB (0.47) LMNAHTTSMN1; SMN2ALDH1A1MAPT
SCHEMBL11224229 0.80 ROCK2 (0.49) AURKATTKAURKBINCENPPDGFRB
SCHEMBL11182349 0.79 AURKA (0.53) AURKATTKAURKBINCENPLMNA
SCHEMBL11235044 0.79 AURKA (0.47) AURKATTKAURKBINCENPROCK2
SCHEMBL11336666 0.77 AURKA (0.45) AURKATTKAURKBINCENPLMNA
Water SCHEMBL11225673 0.76 AURKA (0.44) AURKATTKAURKBINCENPLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4309537-A Production of imidazo[4,5-b]pyridin-2-ones or thiones STERLING DRUG INC. (US) 1982-01-05 US disclosed
US-4297360-A 5-(Pyridinyl)pyridine-2,3-diamines, preparation thereof and their cardiotonic use STERLING DRUG INC. (US) 1981-10-27 US disclosed
US-4294837-A 1,3-Dihydro-6-(pyridinyl)-2H-imidazo[4,5-b]pyridin-2-ones and -imidazo[4,5-b]pyridine-2-thiones and their cardiotonic use STERLING DRUG INC. (US) 1981-10-13 US disclosed
US-4276293-A Compositions and their preparation STERLING DRUG INC. (US) 1981-06-30 US disclosed