SCHEMBL11240971

SCHEMBL11240971

CC(C)(C)c1[nH]c(=O)c(Br)cc1-c1ccncc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 11/20 0.43
PDE3A Q14432 11/20 0.43
KDM4E B2RXH2 1/20 0.43
PDE5A O76074 1/20 0.43
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
PTGS1 P23219 1/20 0.43
PDE4A P27815 1/20 0.43
CYP2C19 P33261 1/20 0.43
BLM P54132 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
AURKB Q96GD4 1/20 0.43
INCENP Q9NQS7 1/20 0.43
HSD17B1 P14061 2/20 0.38
HSD17B2 P37059 2/20 0.38
GCGR P47871 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11238702 0.82 PDE3B (0.66) PDE3BPDE3AKDM4EPDE5ALMNA
SCHEMBL11234713 0.80 PDE3B (0.67) PDE3BPDE3AKDM4EPDE5ALMNA
SCHEMBL11226409 0.79 PDE3A (0.70) PDE3BPDE3AKDM4EPDE5ALMNA
SCHEMBL11237595 0.79 PDE3B (0.42) PDE3BPDE3AKDM4EPDE5ALMNA
SCHEMBL11231155 0.78 HSD17B1 (0.44) PDE3BPDE3AKDM4EPDE5ALMNA
SCHEMBL11227017 0.78 HSD17B1 (0.42) PDE3BPDE3AKDM4EPDE5ALMNA
SCHEMBL11238495 0.77 PDE3B (0.40) PDE3BPDE3AKDM4EPDE5ALMNA
SCHEMBL11239860 0.77 CDC7 (0.48) PDE3BPDE3AAURKBINCENPHSD17B1
SCHEMBL11236260 0.76 PDE3B (0.43) PDE3BPDE3AKDM4EPDE5ALMNA
SCHEMBL11236105 0.75 CYP46A1 (0.51) PDE3BPDE3AKDM4EPDE5ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4365065-A 1-(Pyridinyl)-2-(dimethylamino)ethenyl lower-alkyl ketones STERLING DRUG INC. (US) 1982-12-21 US disclosed
US-4313951-A 3-Substituted-6-(lower-alkyl)-5-(pyridinyl)-2(1H)-pyridinones, their cardiotonic use and intermediates therefor STERLING DRUG INC. (US) 1982-02-02 US disclosed