SCHEMBL1124201

SCHEMBL1124201

NC(=O)/C(=C\c1ccc(C(F)(F)F)cc1)Cc1ccc(N2CCOCC2)nc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.52
MAPT P10636 2/20 0.52
STAT3 P40763 1/20 0.52
AOC3 Q16853 2/20 0.50
KDM4E B2RXH2 1/20 0.44
ABL1 P00519 1/20 0.44
LMNA P02545 1/20 0.44
HIF1A Q16665 2/20 0.43
EPAS1 Q99814 2/20 0.43
FPR1 P21462 1/20 0.41
FPR2 P25090 1/20 0.41
TLR7 Q9NYK1 1/20 0.41
MCHR1 Q99705 1/20 0.40
HPGD P15428 1/20 0.40
ALDH1A1 P00352 1/20 0.40
DGAT1 O75907 1/20 0.39
SOAT1 P35610 1/20 0.39
KCNH2 Q12809 1/20 0.39
HPGDS O60760 1/20 0.39
HSD11B1 P28845 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1124207 1.00 SMN1; SMN2 (0.52) SMN1; SMN2MAPTSTAT3AOC3KDM4E
SCHEMBL1124174 0.87 AOC3 (0.50) SMN1; SMN2MAPTAOC3KDM4ELMNA
SCHEMBL1124168 0.87 AOC3 (0.50) SMN1; SMN2MAPTAOC3KDM4ELMNA
SCHEMBL2338224 0.86 AKR1C3 (0.50) SMN1; SMN2MAPTLMNAHIF1AEPAS1
SCHEMBL2338228 0.86 AKR1C3 (0.50) SMN1; SMN2MAPTLMNAHIF1AEPAS1
SCHEMBL1124204 0.76 SMN1; SMN2 (0.53) SMN1; SMN2MAPTSTAT3AOC3LMNA
SCHEMBL1124111 0.75 AOC3 (0.60) SMN1; SMN2MAPTAOC3KDM4ELMNA
SCHEMBL23683819 0.72 AOC3 (0.62) SMN1; SMN2MAPTAOC3KDM4ELMNA
SCHEMBL30475671 0.72 AOC3 (0.62) SMN1; SMN2MAPTAOC3KDM4ELMNA
SCHEMBL29959269 0.72 MAPT (0.62) SMN1; SMN2MAPTSTAT3AOC3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2282996-A1 TETRAHYDROISOQUINOLINES AS ANTIMALARIAL AGENTS Actelion Pharmaceuticals Ltd. (CH) 2011-02-16 EP claimed
EP-2282996-A1 TETRAHYDROISOQUINOLINES AS ANTIMALARIAL AGENTS Actelion Pharmaceuticals Ltd. (CH) 2011-02-16 EP disclosed