SCHEMBL1124168

SCHEMBL1124168

Cc1ccc(/C=C(/Cc2ccc(N3CCOCC3)nc2)C(N)=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.50
MAPT P10636 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP2C19 P33261 1/20 0.48
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
GAA P10253 4/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
WNT3A P56704 2/20 0.42
ALDH1A1 P00352 5/20 0.42
CACNA1H O95180 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
KDM4E B2RXH2 3/20 0.40
HSD17B10 Q99714 3/20 0.40
HPGD P15428 2/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
RECQL P46063 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1124174 1.00 AOC3 (0.50) AOC3MAPTCYP1A2CYP2C19CYP11B1
SCHEMBL1124207 0.87 SMN1; SMN2 (0.52) AOC3MAPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL1124201 0.87 SMN1; SMN2 (0.52) AOC3MAPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL1124111 0.77 AOC3 (0.60) AOC3MAPTCYP1A2CYP2C19CYP11B1
SCHEMBL23683819 0.74 AOC3 (0.62) AOC3MAPTCYP1A2CYP2C19CYP11B1
SCHEMBL30475671 0.74 AOC3 (0.62) AOC3MAPTCYP1A2CYP2C19CYP11B1
SCHEMBL1124170 0.74 SMN1; SMN2 (0.62) AOC3MAPTCYP1A2CYP2C19CYP11B1
Hydrochloric Acid SCHEMBL20424596 0.73 AOC3 (0.60) AOC3MAPTCYP1A2CYP2C19CYP11B1
SCHEMBL20424591 0.73 AOC3 (0.60) AOC3MAPTCYP1A2CYP2C19CYP11B1
SCHEMBL2338228 0.71 AKR1C3 (0.50) MAPTKMT2AMEN1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2282996-A1 TETRAHYDROISOQUINOLINES AS ANTIMALARIAL AGENTS Actelion Pharmaceuticals Ltd. (CH) 2011-02-16 EP claimed
EP-2282996-A1 TETRAHYDROISOQUINOLINES AS ANTIMALARIAL AGENTS Actelion Pharmaceuticals Ltd. (CH) 2011-02-16 EP disclosed