SCHEMBL11243017

SCHEMBL11243017

C[C@@H]1C[C@H]2[C@@H]3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(Br)[C@@H](O)C[C@]2(C)[C@H]1C(=O)COC(=O)C(C)(C)C

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 10/20 0.80
AR P10275 9/20 0.80
HIF1A Q16665 9/20 0.80
CYP3A4 P08684 6/20 0.80
ADORA3 P0DMS8 4/20 0.80
NR1I2 O75469 3/20 0.61
HTR2B P41595 1/20 0.61
NR3C1 P04150 5/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
CHRM1 P11229 3/20 0.47
LMNA P02545 3/20 0.47
ABCB11 O95342 2/20 0.47
ADRA1A P35348 2/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A3 Q01959 1/20 0.43
KCNH2 Q12809 1/20 0.43
ALDH1A1 P00352 3/20 0.42
CYP1A2 P05177 1/20 0.42
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22171576 0.90 PGR (0.83) PGRARHIF1ACYP3A4ADORA3
Clocortolone Pivalate SCHEMBL10052573 0.89 PGR (1.00) PGRARHIF1ACYP3A4ADORA3
Diflucortolone Pivalate SCHEMBL668257 0.89 PGR (0.81) PGRARHIF1ACYP3A4ADORA3
Clocortolone Pivalate SCHEMBL32668843 0.89 PGR (1.00) PGRARHIF1ACYP3A4ADORA3
Clocortolone Pivalate SCHEMBL5120 0.89 PGR (1.00) PGRARHIF1ACYP3A4ADORA3
Clocortolone Pivalate SCHEMBL6834795 0.89 PGR (1.00) PGRARHIF1ACYP3A4ADORA3
Clocortolone Pivalate SCHEMBL13423591 0.89 PGR (1.00) PGRARHIF1ACYP3A4ADORA3
Diflucortolone Pivalate SCHEMBL668256 0.89 PGR (0.81) PGRARHIF1ACYP3A4ADORA3
SCHEMBL11684094 0.86 PGR (0.61) PGRARHIF1ACYP3A4ADORA3
SCHEMBL11684088 0.86 PGR (0.61) PGRARHIF1ACYP3A4ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4315866-A Process for preparing 11-keto steroids SCHERING, A.G. (DE) 1982-02-16 US disclosed
EP-0030368-A1 Process for the preparation of 11-keto steroids SCHERING AKTIENGESELLSCHAFT (DE) 1981-06-17 EP disclosed