SCHEMBL11243052

SCHEMBL11243052

CC1(c2ccccc2)CC(=O)N(c2ccncc2)C1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 3/20 0.46
BACE1 P56817 6/20 0.46
BACE2 Q9Y5Z0 3/20 0.46
AR P10275 1/20 0.45
CYP19A1 P11511 1/20 0.43
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CTSD P07339 1/20 0.39
ALDH1A1 P00352 3/20 0.39
BCHE P06276 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
THPO P40225 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29116647 0.74 CYP19A1 (0.50) GRM4BACE1BACE2CYP19A1MEN1
SCHEMBL11480980 0.74 POLB (0.57) ARMEN1KMT2AALDH1A1BCHE
Methsuximide SCHEMBL34852 0.73 CYP19A1 (0.70) GRM4BACE1BACE2CYP19A1MEN1
Methsuximide SCHEMBL34853 0.73 CYP19A1 (0.70) GRM4BACE1BACE2CYP19A1MEN1
SCHEMBL10855612 0.71 ALDH1A1 (0.51) BACE1ARMEN1KMT2AALDH1A1
SCHEMBL14037658 0.69 CYP19A1 (0.47) BACE1BACE2CYP19A1CYP2C19LMNA
SCHEMBL11249870 0.69 ALDH1A1 (0.43) GRM4ARALDH1A1BCHESMN1; SMN2
SCHEMBL13684394 0.69 CYP19A1 (0.44) GRM4BACE1CYP19A1MEN1KMT2A
SCHEMBL11930003 0.69 CYP19A1 (0.44) GRM4BACE1CYP19A1MEN1KMT2A
SCHEMBL6055400 0.68 ALDH1A1 (0.50) BACE1MEN1KMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4309541-A CHEMICAL INTERMEDIATES TO QUINAZOLINE HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1982-01-05 US disclosed
US-4255429-A HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1981-03-10 US disclosed