SCHEMBL11243987

SCHEMBL11243987

O=C1CCCC(=O)C1c1c([N+](=O)[O-])cccc1C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HPD P32754 2/20 0.44
ALDH1A1 P00352 2/20 0.39
MAPT P10636 1/20 0.39
TNF P01375 1/20 0.38
IL6 P05231 1/20 0.38
PNMT P11086 1/20 0.35
TDP1 Q9NUW8 2/20 0.35
CA1 P00915 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11222751 0.78 TSHR (0.49) ALDH1A1MAPTTDP1
SCHEMBL11226368 0.78 ALDH1A1 (0.41) ALDH1A1MAPTTDP1
SCHEMBL30152700 0.71 ALDH1A1 (0.46) ALDH1A1MAPTTDP1
SCHEMBL1768922 0.71 ALDH1A1 (0.46) ALDH1A1MAPTTDP1
SCHEMBL18863552 0.70 ALDH1A1 (0.43) ALDH1A1TDP1
SCHEMBL1999849 0.69 ALDH1A1 (0.50) ALDH1A1TDP1
SCHEMBL30627320 0.69 ALDH1A1 (0.50) ALDH1A1TDP1
SCHEMBL1995565 0.69 TDP1 (0.47) ALDH1A1TDP1
SCHEMBL1459395 0.69 TSHR (0.53) ALDH1A1TDP1
SCHEMBL6515 0.69 TDP1 (0.47) ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0007243-B1 2-ARYL-1,3-CYCLOHEXANEDIONE COMPOUNDS AND ALKALI METAL SALTS, AMMONIUM SALTS AND ENOL ESTERS THEREOF, COMPOSITION AND METHOD OF CONTROLLING ACARINA ECTOPARASITES ON WARMBLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1982-11-17 EP disclosed
US-4257858-A REACTING A CYCLOHEXA-1,3-DIONE-2-DIAZIDE WITH AN ARYL COMPOUND UNION CARBIDE CORPORATION (US) 1981-03-24 US disclosed
US-4256658-A CYCLIZATION, BASIC CATALYST UNION CARBIDE CORPORATION (US) 1981-03-17 US disclosed
US-4256657-A CYCLIZATION, ACID CATALYST UNION CARBIDE CORPORATION (US) 1981-03-17 US disclosed
US-4209532-A Biocidal 2-aryl-1,3-cyclohexane dione compounds and alkali metal and ammonium salts thereof UNION CARBIDE CORPORATION (US) 1980-06-24 US disclosed
EP-0007243-A1 2-Aryl-1,3-cyclohexanedione compounds and alkali metal salts, ammonium salts and enol esters thereof, composition and method of controlling acarina ectoparasites on warmblooded animals UNION CARBIDE CORPORATION (US) 1980-01-23 EP disclosed
US-4175135-A Method of controlling acarina ectoparasites on warmblooded animals by orally administering to the animal an ectoparasitically effective amount of a 2-aryl-1,3-cyclohexanedione compound, and alkali metal salts, ammonium salts and enol esters thereof UNION CARBIDE CORPORATION (US) 1979-11-20 US disclosed