SCHEMBL11246437

SCHEMBL11246437

COC(=O)C1Cc2c([nH]c3ccccc23)C(c2ccc(N(C)C)cc2)N1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 2/20 0.78
PDE5A O76074 5/20 0.70
KDM4E B2RXH2 3/20 0.65
TSHR P16473 2/20 0.65
HSD17B10 Q99714 2/20 0.65
HTT P42858 1/20 0.65
MEN1 O00255 3/20 0.62
KMT2A Q03164 3/20 0.62
CYP2D6 P10635 3/20 0.60
MAPK1 P28482 1/20 0.60
ALDH1A1 P00352 3/20 0.57
ALOX12 P18054 1/20 0.57
CYP2C19 P33261 2/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
CYP1A2 P05177 1/20 0.53
GAA P10253 1/20 0.53
MAPT P10636 1/20 0.53
CYP2C9 P11712 1/20 0.53
HPGD P15428 1/20 0.53
ALOX15 P16050 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1921528 0.89 CCKBR (0.85) CCKBRPDE5AKDM4ETSHRHSD17B10
SCHEMBL4600163 0.89 CCKBR (0.85) CCKBRPDE5AKDM4ETSHRHSD17B10
SCHEMBL1921583 0.89 CCKBR (0.85) CCKBRPDE5AKDM4ETSHRHSD17B10
SCHEMBL16489366 0.89 CCKBR (0.85) CCKBRPDE5AKDM4ETSHRHSD17B10
SCHEMBL13402875 0.89 CCKBR (0.85) CCKBRPDE5AKDM4ETSHRHSD17B10
SCHEMBL17760646 0.89 CCKBR (0.85) CCKBRPDE5AKDM4ETSHRHSD17B10
SCHEMBL1921626 0.89 KDM4E (0.66) CCKBRPDE5AKDM4ETSHRHSD17B10
SCHEMBL21309527 0.88 CCKBR (0.83) CCKBRPDE5AKDM4ETSHRHSD17B10
SCHEMBL18531899 0.88 CCKBR (0.83) CCKBRPDE5AKDM4ETSHRHSD17B10
SCHEMBL1520461 0.88 CCKBR (1.00) CCKBRPDE5AKDM4ETSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4336260-A Method and compositions using 1-aryl-1,2,3,4-tetrahydro-β-carboline-3-carboxylic acid for treating depression THE DOW CHEMICAL COMPANY (US) 1982-06-22 US disclosed