SCHEMBL11246552

SCHEMBL11246552

COc1cccc2c1CCC(CC#N)C2=O

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.61
KDM4E B2RXH2 1/20 0.52
LMNA P02545 1/20 0.52
POLB P06746 1/20 0.52
MAPT P10636 1/20 0.52
ACHE P22303 1/20 0.50
HTR2C P28335 2/20 0.45
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
DRD2 P14416 5/20 0.39
DRD3 P35462 3/20 0.39
DRD4 P21917 3/20 0.39
HTR2A P28223 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15700133 0.83 CYP19A1 (0.67) CYP19A1KDM4ELMNAPOLBMAPT
SCHEMBL31028062 0.81 HTR1A (0.47) CYP19A1DRD2DRD3DRD4
SCHEMBL8673224 0.81 CYP19A1 (0.60) CYP19A1KDM4ELMNAPOLBMAPT
SCHEMBL8875326 0.80 CYP19A1 (0.62) CYP19A1KDM4ELMNAPOLBMAPT
SCHEMBL3822324 0.80 CYP19A1 (0.62) CYP19A1KDM4ELMNAPOLBMAPT
SCHEMBL9361537 0.80 MAPT (0.59) CYP19A1KDM4ELMNAPOLBMAPT
SCHEMBL9343214 0.79 CYP19A1 (0.61) CYP19A1KDM4ELMNAPOLBMAPT
Hydrochloric Acid SCHEMBL5459542 0.79 CYP19A1 (0.61) CYP19A1KDM4ELMNAPOLBMAPT
SCHEMBL8671806 0.79 CYP19A1 (0.58) CYP19A1KDM4ELMNAPOLBMAPT
SCHEMBL8671801 0.79 CYP19A1 (0.58) CYP19A1KDM4ELMNAPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4309345-A POTASSIUM-SPARING DIURETICS CIBA-GEIGY CORPORATION (US) 1982-01-05 US disclosed
US-4173633-A DIURETICS CIBA-GEIGY CORPORATION (US) 1979-11-06 US disclosed