SCHEMBL11247683

SCHEMBL11247683

CC(=O)Nc1cc2c(cnn2C(C)=O)cc1C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.50
AURKA O14965 1/20 0.50
DAPK3 O43293 1/20 0.50
CSNK1A1 P48729 1/20 0.50
GSK3A P49840 1/20 0.50
LIMK1 P53667 1/20 0.50
IKBKE Q14164 1/20 0.50
MAPK14 Q16539 1/20 0.50
TAOK1 Q7L7X3 1/20 0.50
CLK4 Q9HAZ1 1/20 0.50
DYRK1B Q9Y463 1/20 0.50
KMT2A Q03164 3/20 0.45
MAPT P10636 3/20 0.44
NPC1 O15118 8/20 0.42
RAB9A P51151 7/20 0.42
ALDH1A1 P00352 4/20 0.41
HPGD P15428 1/20 0.41
MEN1 O00255 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11257612 0.82 CHEK1 (0.48) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL21796520 0.80 CHEK1 (0.54) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL21796872 0.78 IKBKE (0.53) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL836744 0.75 CHEK1 (0.53) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL1542059 0.75 IKBKE (0.53) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL11485102 0.74 CREBBP (0.56) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL5413013 0.74 CHEK1 (0.48) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL21797005 0.72 CHEK1 (0.47) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL26053980 0.72 CHEK1 (0.57) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL29819513 0.72 ALDH1A1 (0.58) KMT2AMAPTNPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4352931-A Lin-benzoaminopurinols SIEGFRIED AKTIENGESELLSCHAFT (CH) 1982-10-05 US disclosed
EP-0040872-A1 Pyrazolo-quinazoline derivatives and methods of producing such derivatives SIEGFRIED AKTIENGESELLSCHAFT (CH) 1981-12-02 EP disclosed