SCHEMBL11248010

SCHEMBL11248010

CNC(=S)Nc1cccc(-c2csc(NC(=N)N)n2)c1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIRT5 Q9NXA8 7/20 0.52
NPC1 O15118 5/20 0.51
RAB9A P51151 5/20 0.51
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
JAK2 O60674 1/20 0.51
MAPT P10636 6/20 0.49
GAA P10253 2/20 0.49
NPSR1 Q6W5P4 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.47
ALDH1A1 P00352 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
NFKB1 P19838 2/20 0.46
NFKB2 Q00653 2/20 0.46
RELA Q04206 2/20 0.46
ABL1 P00519 2/20 0.46
KDM4E B2RXH2 1/20 0.44
HDAC3 O15379 1/20 0.44
NCOR2 Q9Y618 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL11247631 0.95 SIRT5 (0.55) SIRT5NPC1RAB9AMEN1KMT2A
SCHEMBL11246181 0.88 MAPT (0.53) SIRT5NPC1RAB9AMEN1KMT2A
SCHEMBL11239265 0.88 MAPT (0.57) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL3608636 0.87 MAPT (0.51) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL11248461 0.86 MAPT (0.55) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL3612694 0.84 MAPT (0.67) SIRT5NPC1RAB9AMEN1KMT2A
SCHEMBL10675056 0.83 MAPT (0.50) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL11253950 0.82 MAPT (0.64) SIRT5NPC1RAB9AMEN1KMT2A
SCHEMBL11245298 0.82 MAPT (0.45) SIRT5NPC1RAB9AMEN1KMT2A
SCHEMBL11245292 0.82 MAPT (0.45) SIRT5NPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4315009-A Antisecretory guanidine derivatives and pharmaceutical compositions containing them IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1982-02-09 US disclosed
EP-0003640-A2 Antisecretory guanidine derivatives, processes for their manufacture and pharmaceutical compositions containing them IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1979-08-22 EP disclosed