SCHEMBL11248967

SCHEMBL11248967

CN(c1ccc(C(=O)O)cc1)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.42
MEN1 O00255 1/20 0.42
POLB P06746 1/20 0.42
KMT2A Q03164 1/20 0.42
NR1H3 Q13133 2/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
SRD5A2 P31213 4/20 0.39
HPGD P15428 3/20 0.38
ALDH1A1 P00352 3/20 0.37
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NR1H2 P55055 1/20 0.36
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36
MAPT P10636 1/20 0.35
RAB9A P51151 2/20 0.35
CA12 O43570 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11247704 1.00 NPC1 (0.42) NPC1MEN1POLBKMT2ANR1H3
SCHEMBL16730055 0.86 NPC1 (0.47) NPC1MEN1POLBKMT2ANR1H3
SCHEMBL11255588 0.80 CA12 (0.46) NPC1MEN1POLBKMT2ATP53
SCHEMBL16730050 0.79 NPC1 (0.50) NPC1MEN1POLBKMT2ATP53
SCHEMBL6792995 0.79 MEN1 (0.37) MEN1KMT2ANR1H3TSHRALDH1A1
Perflubutane SCHEMBL28930534 0.78 TSHR (0.63) TP53TSHRSRD5A2HPGDALDH1A1
SCHEMBL11317352 0.75 CYP2A6 (0.48) ALDH1A1TYR
SCHEMBL16730046 0.73 NPC1 (0.52) NPC1MEN1POLBKMT2ATP53
Perflubutane SCHEMBL28615208 0.70 TSHR (0.67) POLBTP53TSHRSRD5A2ALDH1A1
SCHEMBL2058690 0.70 SRD5A2 (0.53) MEN1KMT2ATP53TSHRSRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4310545-A Hypolipidemic and antiatherosclerotic 4-(polyfluoroalkylamino) phenyl compounds AMERICAN CYANAMID COMPANY (US) 1982-01-12 US claimed
US-4318914-A Hypolipidemic and antiatherosclerotic 4-(polyfluoro-alkylamino)phenyl compounds AMERICAN CYANAMID COMPANY (US) 1982-03-09 US disclosed
US-4310545-A Hypolipidemic and antiatherosclerotic 4-(polyfluoroalkylamino) phenyl compounds AMERICAN CYANAMID COMPANY (US) 1982-01-12 US disclosed
US-4305959-A Hypolipidemic and antiatherosclerotic 4-(polyfluoro-alkylamino)phenyl compounds AMERICAN CYANAMID COMPANY (US) 1981-12-15 US disclosed
US-4205085-A Hypolipidemic and antiatherosclerotic 4-(polyfluoroalkylamino)phenyl compounds AMERICAN CYANAMID COMPANY (US) 1980-05-27 US disclosed
EP-0003663-A2 Amino-substituted phenyl and heteroaryl compounds, process for their preparation and pharmaceutical compositions containing them AMERICAN CYANAMID COMPANY (US) 1979-08-22 EP disclosed