Bromide

Bromide

SCHEMBL11249987

Br.O=C1c2cc(Cl)ccc2Oc2ccccc2C12CCN(CC1CC1)CC2

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 known ✓ Q99720 5/20 0.38
HRH1 P35367 2/20 0.55
HTR2A P28223 1/20 0.55
OPRL1 P41146 12/20 0.43
OPRM1 P35372 8/20 0.43
OPRK1 P41145 6/20 0.43
DRD2 P14416 3/20 0.37
PGR P06401 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11244394 0.99 HRH1 (0.56) HRH1HTR2AOPRL1OPRM1OPRK1
Bromide SCHEMBL11255909 0.88 OPRL1 (0.48) HRH1HTR2AOPRL1OPRM1OPRK1
Bromide SCHEMBL11482097 0.86 HTR2A (0.53) HRH1HTR2AOPRM1OPRK1SIGMAR1
SCHEMBL11315886 0.85 HTR2A (0.54) HRH1HTR2AOPRM1OPRK1SIGMAR1
Bromide SCHEMBL11245480 0.84 HTR2A (0.52) HRH1HTR2AOPRM1OPRK1SIGMAR1
Bromide SCHEMBL11318175 0.84 HTR2A (0.54) HRH1HTR2AOPRM1OPRK1SIGMAR1
Bromide SCHEMBL11475283 0.84 HRH1 (0.51) HRH1HTR2AOPRM1OPRK1SIGMAR1
Bromide SCHEMBL11473841 0.83 HRH1 (0.56) HRH1HTR2AOPRM1OPRK1DRD2
SCHEMBL11490180 0.82 HTR2A (0.54) HRH1HTR2AOPRM1OPRK1SIGMAR1
SCHEMBL11479513 0.82 HTR2A (0.53) HRH1HTR2AOPRM1SIGMAR1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0016261-B1 SPIRO(DIBENZ(B,F)OXEPIN-PIPERIDINES) AND METHODS OF PREPARING SAME HOECHST AKTIENGESELLSCHAFT (DE) 1982-12-29 EP disclosed
US-4198418-A ANALGESICS, TRANQUILIZERS, ANTICONVULSANTS AMERICAN HOECHST CORPORATION (US) 1980-04-15 US disclosed