SCHEMBL11250593

SCHEMBL11250593

COC(=O)COc1cccc(CC(C)NCC(O)c2ccc(O)c(CO)c2)c1

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 18/20 0.62
ADRB1 P08588 2/20 0.61
ADRB3 P13945 2/20 0.61
GLA P06280 1/20 0.61
ADRA1D P25100 1/20 0.50
ADRA1A P35348 1/20 0.50
ADRA1B P35368 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11249876 0.90 ADRB2 (0.69) ADRB2ADRB1ADRB3GLAADRA1D
SCHEMBL4256482 0.85 ADRB2 (0.67) ADRB2ADRB1ADRB3GLA
SCHEMBL10895573 0.85 ADRB3 (0.83) ADRB2ADRB1ADRB3GLAADRA1D
SCHEMBL10661675 0.83 ADRB2 (0.66) ADRB2ADRB1ADRB3
SCHEMBL4386774 0.83 ADRB2 (0.66) ADRB2ADRB1ADRB3
SCHEMBL4386778 0.83 ADRB2 (0.66) ADRB2ADRB1ADRB3
SCHEMBL14422857 0.81 ADRB2 (0.61) ADRB2ADRB1ADRB3GLAADRA1A
SCHEMBL4384732 0.81 ADRB2 (0.71) ADRB2ADRB1ADRB3
SCHEMBL4256480 0.81 ADRB2 (0.74) ADRB2
SCHEMBL14422860 0.81 ADRB2 (0.80) ADRB2ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4338333-A ANTIOBESITY, HYPOGLYCEMIC BEECHAM GROUP LIMITED (GB) 1982-07-06 US claimed
US-4338333-A ANTIOBESITY, HYPOGLYCEMIC BEECHAM GROUP LIMITED (GB) 1982-07-06 US disclosed
EP-0023385-A1 Ethanamine derivatives, their preparation and use in pharmaceutical compositions BEECHAM GROUP PLC (GB) 1981-02-04 EP disclosed