SCHEMBL11250696

SCHEMBL11250696

O=C(NCCNCc1ccccc1)[C@@H]1CCCN1C(=O)Cc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 3/20 0.59
POLB P06746 2/20 0.55
ITGB1 P05556 4/20 0.55
ITGA4 P13612 4/20 0.55
ALDH1A1 P00352 2/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2C9 P11712 1/20 0.55
PKM P14618 1/20 0.55
CYP2C19 P33261 1/20 0.55
F2 P00734 1/20 0.52
NPC1 O15118 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11250683 1.00 FKBP1A (0.59) FKBP1APOLBITGB1ITGA4ALDH1A1
SCHEMBL11250707 1.00 FKBP1A (0.59) FKBP1APOLBITGB1ITGA4ALDH1A1
Bromide SCHEMBL11247303 0.99 FKBP1A (0.58) FKBP1APOLBITGB1ITGA4ALDH1A1
Bromide SCHEMBL11247292 0.99 FKBP1A (0.58) FKBP1APOLBITGB1ITGA4ALDH1A1
Bromide SCHEMBL11247297 0.99 FKBP1A (0.58) FKBP1APOLBITGB1ITGA4ALDH1A1
SCHEMBL9139680 0.86 ITGB1 (0.61) FKBP1APOLBITGB1ITGA4ALDH1A1
SCHEMBL11248906 0.86 FKBP1A (0.57) FKBP1APOLBITGB1ITGA4ALDH1A1
SCHEMBL11248915 0.86 FKBP1A (0.57) FKBP1APOLBITGB1ITGA4ALDH1A1
SCHEMBL11248907 0.86 FKBP1A (0.57) FKBP1APOLBITGB1ITGA4ALDH1A1
SCHEMBL6352517 0.84 ITGB1 (0.55) FKBP1APOLBITGB1ITGA4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0019411-B1 1-PHENYL-2-AMINOETHANOL DERIVATIVES, PROCESSES FOR THEIR MANUFACTURE AND PHARMACEUTICAL COMPOSITIONS THEREOF IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-12-22 EP disclosed
US-4323575-A TOPICAL ANTIINFLAMMATORY AGENTS IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1982-04-06 US disclosed
EP-0019411-A1 1-Phenyl-2-aminoethanol derivatives, processes for their manufacture and pharmaceutical compositions thereof IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1980-11-26 EP disclosed