Peraclopone

Peraclopone

SCHEMBL11255181

OC(CO/N=C\c1ccc(Cl)cc1)CN1CCN(c2ccccc2Cl)CC1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.53
MAPT P10636 3/20 0.53
MAPK1 P28482 2/20 0.53
NPSR1 Q6W5P4 2/20 0.53
HTR7 P34969 1/20 0.51
HTT P42858 5/20 0.50
ALDH1A1 P00352 2/20 0.50
GAA P10253 2/20 0.50
KMT2A Q03164 2/20 0.48
USP2 O75604 3/20 0.47
MEN1 O00255 1/20 0.47
HSP90AB1 P08238 1/20 0.47
DRD2 P14416 2/20 0.46
DRD3 P35462 2/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
TSHR P16473 1/20 0.46
IGF1R P08069 1/20 0.46
RAB9A P51151 1/20 0.44
RECQL P46063 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Peraclopone SCHEMBL11255188 1.00 KDM4E (0.53) KDM4EMAPTMAPK1NPSR1HTR7
Peraclopone SCHEMBL2110307 1.00 KDM4E (0.53) KDM4EMAPTMAPK1NPSR1HTR7
Peraclopone SCHEMBL11266970 0.99 KDM4E (0.52) KDM4EMAPTMAPK1NPSR1HTR7
Peraclopone SCHEMBL11251964 0.99 KDM4E (0.52) KDM4EMAPTMAPK1NPSR1HTR7
Peraclopone SCHEMBL11266972 0.99 KDM4E (0.52) KDM4EMAPTMAPK1NPSR1HTR7
Peraclopone SCHEMBL11251959 0.99 KDM4E (0.52) KDM4EMAPTMAPK1NPSR1HTR7
SCHEMBL11255248 0.83 MAPT (0.52) MAPTMAPK1NPSR1HTTGAA
SCHEMBL11255243 0.83 MAPT (0.52) MAPTMAPK1NPSR1HTTGAA
Hydrochloric Acid SCHEMBL11247700 0.78 TSHR (0.57) KDM4EMAPTMAPK1HTR7ALDH1A1
Hydrochloric Acid SCHEMBL11247706 0.78 TSHR (0.57) KDM4EMAPTMAPK1HTR7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4358450-A FOR DECREASING BLOOD CHOLESTEROL HOECHST AKTIENGESELLSCHAFT (DE) 1982-11-09 US claimed
US-4358450-A FOR DECREASING BLOOD CHOLESTEROL HOECHST AKTIENGESELLSCHAFT (DE) 1982-11-09 US disclosed