SCHEMBL11261590

SCHEMBL11261590

Clc1cccc2c1CC1(CCNCC1)O2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.49
HTR2B P41595 3/20 0.49
OPRD1 P41143 4/20 0.41
PNMT P11086 1/20 0.37
HTR5A P47898 2/20 0.34
HTR1A P08908 1/20 0.34
HTR1D P28221 1/20 0.34
HTR2A P28223 1/20 0.34
HTR7 P34969 1/20 0.34
HTR3A P46098 1/20 0.34
KCNH2 Q12809 3/20 0.33
HDAC3 O15379 2/20 0.33
HDAC4 P56524 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC7 Q8WUI4 2/20 0.33
HDAC2 Q92769 2/20 0.33
HDAC10 Q969S8 2/20 0.33
HDAC11 Q96DB2 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1589928 0.86 HTR2C (0.48) HTR2CHTR2BOPRD1PNMTHTR2A
Hydrochloric Acid SCHEMBL1591008 0.84 HTR2C (0.47) HTR2CHTR2BOPRD1PNMTHTR2A
SCHEMBL31515333 0.81 OPRD1 (0.41) HTR2CHTR2BOPRD1KCNH2HDAC3
SCHEMBL1590677 0.79 HTR2C (0.45) HTR2CHTR2BOPRD1HDAC3HDAC4
Hydrochloric Acid SCHEMBL3716008 0.78 HTR2C (0.44) HTR2CHTR2BOPRD1HDAC3HDAC4
SCHEMBL24408865 0.75 HTR2C (0.35) HTR2CHTR2BOPRD1HDAC3HDAC4
Hydrochloric Acid SCHEMBL10502304 0.74 HTR2C (0.49) HTR2CHTR2BOPRD1PNMTHTR5A
SCHEMBL231585 0.73 OPRD1 (0.49) HTR2CHTR2BOPRD1HTR2AKCNH2
SCHEMBL24408860 0.72 HTR2C (0.35) HTR2CHTR2BHTR2A
Hydrochloric Acid SCHEMBL10502202 0.71 OPRD1 (0.48) HTR2CHTR2BOPRD1HTR2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0004952-B1 SPIRO-(DIHYDROBENZOFURANPIPERIDINES AND -PYRROLIDINES) AND DERIVATIVES THEREOF, METHODS FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1982-04-07 EP disclosed
US-4166119-A Analgesic and tranquilizing spiro[dihydrobenzofuran]piperidines and pyrrolidines AMERICAN HOECHST CORPORATION (US) 1979-08-28 US disclosed