SCHEMBL11262091

SCHEMBL11262091

COC(=O)C(C)c1ccncc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.57
HPGD P15428 1/20 0.50
KMT2A Q03164 1/20 0.47
PTGS2 P35354 2/20 0.46
PTGS1 P23219 1/20 0.46
CYP17A1 P05093 1/20 0.46
POLB P06746 1/20 0.43
TSHR P16473 1/20 0.43
MT-CO2 P00403 1/20 0.43
ROCK2 O75116 2/20 0.42
ROCK1 Q13464 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
MDM2 Q00987 1/20 0.42
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
LMNA P02545 1/20 0.41
FFAR2 O15552 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12896270 1.00 CYP19A1 (0.57) CYP19A1HPGDKMT2APTGS2PTGS1
SCHEMBL29705753 0.82 ALDH1A1 (0.51) CYP19A1KMT2APTGS2POLBTSHR
SCHEMBL27540323 0.81 CYP19A1 (0.54) CYP19A1PTGS2CYP17A1CYP2C19LMNA
SCHEMBL755729 0.81 CYP19A1 (0.54) CYP19A1HPGDKMT2ACYP17A1POLB
SCHEMBL5537242 0.79 KMT2A (0.67) HPGDKMT2APTGS2PTGS1POLB
SCHEMBL5544986 0.79 KMT2A (0.67) HPGDKMT2APTGS2PTGS1POLB
SCHEMBL12896284 0.79 HPGD (0.53) HPGDKMT2APTGS2PTGS1MT-CO2
SCHEMBL11130803 0.79 HPGD (0.53) HPGDKMT2APTGS2PTGS1MT-CO2
SCHEMBL183940 0.79 KMT2A (0.67) HPGDKMT2APTGS2PTGS1POLB
SCHEMBL9111312 0.79 CYP19A1 (0.50) CYP19A1KMT2APTGS2CYP17A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1027504-C Process for the preparation of imidazolyl-alkenoic acids SMITHKLINE BEECHAM CORP (US) 1995-01-25 CN disclosed
CN-1048038-A IMIDAZOLYL-ALKENOIC ACIDS SMITHKLINE BEECHAM CORP (US) 1990-12-26 CN disclosed
EP-0060144-A2 Cephalosporin antibiotics ELI LILLY AND COMPANY (US) 1982-09-15 EP disclosed
US-4336253-A Cephalosporin antibiotics ELI LILLY AND COMPANY (US) 1982-06-22 US disclosed