SCHEMBL11264323

SCHEMBL11264323

CCc1nccc2c(CC#N)cccc12

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.36
PDE3A Q14432 2/20 0.36
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
TDO2 P48775 1/20 0.32
KDM4D Q6B0I6 1/20 0.32
PDE10A Q9Y233 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11262866 0.88 PDE3B (0.38) PDE3BPDE3AKDM4EALDH1A1HPGD
SCHEMBL11257186 0.84 PDE3B (0.40) PDE3BPDE3AKDM4EALDH1A1HPGD
SCHEMBL22114028 0.83 PDE3B (0.45) PDE3BPDE3AKDM4EALDH1A1TDO2
SCHEMBL11246499 0.83 TDP1 (0.37) KDM4E
SCHEMBL11258743 0.78 ALDH1A1 (0.32) ALDH1A1HPGD
SCHEMBL11257770 0.78
SCHEMBL21617927 0.77 ALDH1A1 (0.45) KDM4EALDH1A1HPGD
SCHEMBL11251945 0.77 CYP3A4 (0.31) ALDH1A1HPGD
SCHEMBL11267998 0.77 ALDH1A1 (0.32) ALDH1A1HPGD
SCHEMBL31583253 0.75 PLAU (0.46) PDE3BPDE3AKDM4EALDH1A1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed