SCHEMBL11264773

SCHEMBL11264773

O=C1CC2(CCCC2)CC(=O)N1c1ccncc1

nearest known ligand 0.69

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.49
BCHE P06276 1/20 0.46
ALDH1A1 P00352 2/20 0.45
AR P10275 1/20 0.41
USP2 O75604 1/20 0.40
CYP3A4 P08684 4/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
TSHR P16473 2/20 0.40
CYP2D6 P10635 1/20 0.40
HTR1A P08908 2/20 0.38
MAPK1 P28482 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
CHKA P35790 1/20 0.38
EP300 Q09472 1/20 0.37
KAT2B Q92831 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11251498 0.98 SMN1; SMN2 (0.47) SMN1; SMN2BCHEALDH1A1ARUSP2
SCHEMBL11253978 0.80 GAA (0.49) SMN1; SMN2ALDH1A1ARHTR1AMAPK1
SCHEMBL11249870 0.79 ALDH1A1 (0.43) SMN1; SMN2BCHEALDH1A1ARUSP2
SCHEMBL13949620 0.79 SMN1; SMN2 (0.57) SMN1; SMN2ALDH1A1HTR1AADRA1AADRA1B
SCHEMBL11480980 0.78 POLB (0.57) SMN1; SMN2BCHEALDH1A1ARUSP2
SCHEMBL4998277 0.76 SMN1; SMN2 (0.43) SMN1; SMN2HTR1AKMT2AADRA1AADRA1B
SCHEMBL11251034 0.75 KMT2A (0.59) SMN1; SMN2BCHEALDH1A1ARUSP2
SCHEMBL11266599 0.74 BCHE (0.58) SMN1; SMN2BCHEALDH1A1ARUSP2
SCHEMBL4763016 0.73 SMN1; SMN2 (0.46) SMN1; SMN2HTR1AMEN1KMT2AADRA1A
SCHEMBL2943787 0.70 ALDH1A1 (0.53) SMN1; SMN2ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4309541-A CHEMICAL INTERMEDIATES TO QUINAZOLINE HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1982-01-05 US disclosed
US-4255429-A HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1981-03-10 US disclosed