SCHEMBL11270913

SCHEMBL11270913

NCCc1cccc2cnccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.55
CYP2D6 P10635 2/20 0.55
LMNA P02545 2/20 0.55
CYP1A2 P05177 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
KDM4E B2RXH2 2/20 0.50
MAPKAPK2 P49137 1/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
PRKD3 O94806 1/20 0.49
TP53 P04637 1/20 0.49
PRKCG P05129 1/20 0.49
PRKCB P05771 1/20 0.49
PRKCA P17252 1/20 0.49
PRKACA P17612 1/20 0.49
NFKB1 P19838 1/20 0.49
PRKACG P22612 1/20 0.49
PRKACB P22694 1/20 0.49
PRKCH P24723 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL263884 0.85 CYP3A4 (0.58) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL30098481 0.85 CYP3A4 (0.58) CYP3A4CYP2D6LMNACYP1A2CYP2C9
Hydrochloric Acid SCHEMBL4783267 0.84 LMNA (0.56) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL6965122 0.82 CYP3A4 (0.50) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL6114531 0.82 KDM4E (0.50) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL27407502 0.82 CYP2D6 (0.50) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL1830568 0.82 KDM4E (0.55) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL6114998 0.79 TRPV1 (0.51) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL14194581 0.79 PRKCH (0.53) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL17028190 0.79 PDE10A (0.44) CYP3A4CYP2D6LMNACYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed