SCHEMBL1127258

SCHEMBL1127258

CCOC(=O)c1c(-c2ccccc2)c(C(=O)OCC)n(CCOC)c1CC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.48
GAA P10253 4/20 0.48
ALDH1A1 P00352 4/20 0.48
KDM4E B2RXH2 4/20 0.48
HPGD P15428 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
LMNA P02545 2/20 0.48
RAB9A P51151 2/20 0.48
NPC1 O15118 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
TSHR P16473 2/20 0.46
HSD17B10 Q99714 2/20 0.45
TDP1 Q9NUW8 1/20 0.44
TP53 P04637 2/20 0.44
GRM6 O15303 1/20 0.44
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1126643 0.88 TSHR (0.54) MAPTGAAALDH1A1KDM4EHPGD
SCHEMBL1126572 0.88 MAPT (0.50) MAPTGAAALDH1A1KDM4EHPGD
SCHEMBL1126660 0.84 MAPT (0.46) MAPTGAAALDH1A1KDM4EHPGD
SCHEMBL1127071 0.83 GRIA2 (0.45) ALDH1A1HPGDLMNATDP1TP53
SCHEMBL1127080 0.83 TSHR (0.55) MAPTGAAALDH1A1KDM4EHPGD
SCHEMBL1991365 0.82 TSHR (0.50) MAPTGAAALDH1A1KDM4EHPGD
SCHEMBL1994935 0.79 TSHR (0.54) MAPTGAAALDH1A1KDM4EHPGD
SCHEMBL1990320 0.78 TSHR (0.48) MAPTGAAALDH1A1KDM4EHPGD
SCHEMBL1126745 0.77 TSHR (0.52) MAPTGAAALDH1A1KDM4EHPGD
SCHEMBL1127099 0.77 TSHR (0.57) MAPTGAAALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-B1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2015-02-25 EP disclosed
EP-2626361-B1 Pyrrole antifungal agents F2G LTD (GB) 2014-10-15 EP disclosed
EP-2626361-A1 Pyrrole antifungal agents F2G Limited (GB) 2013-08-14 EP disclosed
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed